Found 3 Enz. Inhib. hit(s) with Target = 'Transcriptional activator protein LasR' and Ligand = 'BDBM50248862'
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Universidad De Cartagena-Facultad De Ciencias Exactas Y
Curated by ChEMBL
Universidad De Cartagena-Facultad De Ciencias Exactas Y
Curated by ChEMBL
Affinity DataIC50: 5.36E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Universidad De Cartagena-Facultad De Ciencias Exactas Y
Curated by ChEMBL
Universidad De Cartagena-Facultad De Ciencias Exactas Y
Curated by ChEMBL
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Universidad De Cartagena-Facultad De Ciencias Exactas Y
Curated by ChEMBL
Universidad De Cartagena-Facultad De Ciencias Exactas Y
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair