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Found 3 Enz. Inhib. hit(s) with Target = 'Transcriptional activator protein LasR' and Ligand = 'BDBM50248862'
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Universidad De Cartagena-Facultad De Ciencias Exactas Y

Curated by ChEMBL
LigandPNGBDBM50248862(CHEMBL473592 | N-(3-oxo-3-phenylpropanoyl)-L-homos...)
Affinity DataIC50:  5.36E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Universidad De Cartagena-Facultad De Ciencias Exactas Y

Curated by ChEMBL
LigandPNGBDBM50248862(CHEMBL473592 | N-(3-oxo-3-phenylpropanoyl)-L-homos...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Universidad De Cartagena-Facultad De Ciencias Exactas Y

Curated by ChEMBL
LigandPNGBDBM50248862(CHEMBL473592 | N-(3-oxo-3-phenylpropanoyl)-L-homos...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR receptor expressed in Escherichia coli in absence of natural autoinducerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed