Found 3 Enz. Inhib. hit(s) with Target = 'Transcriptional activator protein LasR' and Ligand = 'BDBM50300131'
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Nottingham
Curated by ChEMBL
University Of Nottingham
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Antagonist activity at GFP-fused LasR in Pseudomonas aeruginosa PAO-JP2 co-expressing LVAgfp plasmid by fluorescence assayMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Nottingham
Curated by ChEMBL
University Of Nottingham
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
University Of Nottingham
Curated by ChEMBL
University Of Nottingham
Curated by ChEMBL
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair