Found 2 Enz. Inhib. hit(s) with Target = 'Transcriptional enhancer factor TEF-3' and Ligand = 'BDBM30815'
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Shanghai Institute Of Materia Medica
Curated by ChEMBL
Shanghai Institute Of Materia Medica
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of N-terminal His6-tagged human TEAD4 YAP binding domain (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells assessed redu...More data for this Ligand-Target Pair
TargetTranscriptional enhancer factor TEF-3(Homo sapiens)
Shanghai Institute Of Materia Medica
Curated by ChEMBL
Shanghai Institute Of Materia Medica
Curated by ChEMBL
Affinity DataKd: 4.10E+4nMAssay Description:Binding affinity to N-terminal His6 tagged human TEAD4-YBD (217 to 434 residues) expressed in Escherichia coli C43 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair