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Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM481772'
LigandPNGBDBM481772((R)-3-(2-(4-chlorophenyl)- 2-fluoroethyl)-5-((7-me...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at rat TRPA1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM481772((R)-3-(2-(4-chlorophenyl)- 2-fluoroethyl)-5-((7-me...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human TRPA1 expressed in CHO cells measured by calcium based FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM481772((R)-3-(2-(4-chlorophenyl)- 2-fluoroethyl)-5-((7-me...)
Affinity DataIC50:  34nMAssay Description:The IC50 (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent