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Found 4 Enz. Inhib. hit(s) with Target = 'Transporter' and Ligand = 'BDBM50045824'
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50045824(8-Methyl-2-(3-methyl-[1,2,4]oxadiazol-5-yl)-3-phen...)
Affinity DataIC50:  7.88E+3nMAssay Description:Binding affinity towards norepinephrine transporter by displacement of [3H]nisoxetine radioligand from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50045824(8-Methyl-2-(3-methyl-[1,2,4]oxadiazol-5-yl)-3-phen...)
Affinity DataIC50:  7.88E+3nMAssay Description:Binding affinity towards norepinephrine transporter by displacement of [3H]nisoxetine radioligand from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50045824(8-Methyl-2-(3-methyl-[1,2,4]oxadiazol-5-yl)-3-phen...)
Affinity DataIC50:  3.58E+4nMAssay Description:Binding affinity towards norepinephrine transporter by displacement of [3H]nisoxetine radioligand from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50045824(8-Methyl-2-(3-methyl-[1,2,4]oxadiazol-5-yl)-3-phen...)
Affinity DataIC50:  7.10E+4nMAssay Description:Binding affinity towards norepinephrine transporter by displacement of [3H]nisoxetine radioligand from rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed