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Found 2 Enz. Inhib. hit(s) with Target = 'Tryptase beta-2' and Ligand = 'BDBM16308'
TargetTryptase beta-2(Homo sapiens (Human))
Arris

LigandPNGBDBM16308(2-(isoquinolin-1-yl)-1H-1,3-benzodiazole-6-carboxi...)
Affinity DataKi:  8.80E+3nMAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2(Homo sapiens (Human))
Arris

LigandPNGBDBM16308(2-(isoquinolin-1-yl)-1H-1,3-benzodiazole-6-carboxi...)
Affinity DataKi:  5.45E+4nM ΔG°:  -24.1kJ/molepH: 8.2 T: 2°CAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed