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Found 3 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor' and Ligand = 'BDBM50236697'
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKi:  1.40nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKi:  1.90nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataIC50:  2nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In DepthDetails