Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1 [T315I]/Breakpoint cluster region protein' and Ligand = 'BDBM50591912'
TargetTyrosine-protein kinase ABL1 [T315I]/Breakpoint cluster region protein(Homo sapiens (Human))
Xi'An Jiaotong University
Curated by ChEMBL
Xi'An Jiaotong University
Curated by ChEMBL
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of Bcr-Abl T315I mutant (unknown origin) incubated for 1 hr in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair