Affinity DataIC50: 4.60nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human FRK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Binding constant for FRK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Average Binding Constant for FRK; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Binding constant for FRK kinase domainMore data for this Ligand-Target Pair