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Found
1
Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK2' and Ligand = 'BDBM277755'
Target
Tyrosine-protein kinase JAK2
(Homo sapiens (Human))
Gilead Sciences
US Patent
Ligand
BDBM277755
((R)-methyl 3-(2-cyano-4-(4-((4-(4-(oxetan-3-yl)pip...)
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Affinity Data
IC50: 6.60E+5nM
pH: 7.5
Assay Description:
Enzymatic activity of hJAK2 was measured using a LANCE homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that monitors...
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Target Info
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Ligand Info
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