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Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK2' and Ligand = 'BDBM50466000'
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50466000(CHEMBL4287893)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of JAK2 (unknown origin) preincubated for 20 mins followed by [33P]-ATP addition measured after 2 hrs by filter-binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed