Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase JAK3 [781-1124]' and Ligand = 'BDBM228757'
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Hutchison Medipharma

US Patent
LigandPNGBDBM228757(US10369153, Compound 201 | US9346810, 201)
Affinity DataIC50:  0.550nMT: 2°CAssay Description:JAK1/2/3 kinase assay are performed in vitro using Kit-Tyr 6 Peptide (Invitrogen, Cat. No. PV4122). TYK2 kinase assay are performed in vitro using Z'...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent