Found 7 Enz. Inhib. hit(s) with Target = 'Urokinase-type plasminogen activator' and Ligand = 'BDBM50531925'
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Inhibition of human uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.94E+4nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 354nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataKd: 398nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair