Affinity DataIC50: 372nMAssay Description:Compound was evaluated for OT receptor affinity by displacement of [3H]OT from binding sites in uterine tissue taken from nonlabor pregnant womenMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in CHO cell membranes assessed as inhibition of AVP-induced IP1 accumulation by measur...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human OTR expressed in CHO cell membranes assessed as inhibition of OT-induced IP1 accumulation measured after 1 hr by fluores...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+4nMAssay Description:In vitro for histamine H1 receptor antagonist activity against histamine-induced contractions on isolated guinea pig ileumMore data for this Ligand-Target Pair