TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Induction of bovine serum albumin denaturation incubated for 23 mins by UV-Visible spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of sheep COX-2 by Cayman colorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of sheep COX-2 by Cayman colorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of sheep COX-2 by Cayman colorimetric analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 161nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of ovine COX-1More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 752nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 776nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 791nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of DNA topoisomerase 2 (unknown origin)More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of 5-LOX (unknown origin) by colorimetric analysisMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of 5-LOX (unknown origin) by colorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of recombinant human sPLA2-VMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibition of 5-LOX (unknown origin) by colorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.65E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human SIRT1 expressed in Escherichia coli using Fluor de Lys-SIRT1/2 substrate in presence of NAD+ by fluorescence micropla...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of ovine COX-2More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of recombinant human SIRT1 expressed in Escherichia coli using Fluor de Lys-SIRT1/2 substrate in presence of NAD+ by fluorescence micropla...More data for this Ligand-Target Pair
Affinity DataIC50: 5.77E+3nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hrs by colorimetric analysisMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 7.34E+3nMAssay Description:Inhibition of ovine COX-1More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Prince Sattam Bin Abdulaziz University
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of ovine COX-1More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Mansoura University
Curated by ChEMBL
Mansoura University
Curated by ChEMBL
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of recombinant human SIRT1 expressed in Escherichia coli using Fluor de Lys-SIRT1/2 substrate in presence of NAD+ by fluorescence micropla...More data for this Ligand-Target Pair
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