TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:The compound was tested for its inhibitory activity against beta-mannosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 57nM ΔG°: -10.3kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 72nM ΔG°: -10.1kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 401nM ΔG°: -9.07kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 975nM ΔG°: -8.52kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nM ΔG°: -8.51kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nM ΔG°: -8.30kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nM ΔG°: -8.11kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nM ΔG°: -8.05kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nM ΔG°: -8.05kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nM ΔG°: -8.02kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nM ΔG°: -7.97kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition against Beta-mannosidase in snailMore data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:The compound was tested for its inhibitory activity against beta-mannosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nM ΔG°: -7.03kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nM ΔG°: -6.93kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:The compound was tested for its inhibitory activity against beta-mannosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+4nM ΔG°: -6.61kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition against Beta-mannosidase in snailMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+5nM ΔG°: -4.68kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+6nM ΔG°: -4.25kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
TargetBeta-mannosidase(Homo sapiens (Human))
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
S.E.S.N.A.B., Pole Sciences Et Technologie, Universit�
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMpH: 4.0Assay Description:Inhibition of snail beta mannosidase at pH 4More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+6nM ΔG°: -3.83kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+6nM ΔG°: -3.15kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 9.00E+6nM ΔG°: -2.90kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+7nM ΔG°: -2.78kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+7nM ΔG°: -2.63kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+7nM ΔG°: -2.41kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 2.30E+7nM ΔG°: -2.32kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+7nM ΔG°: -2.10kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: >4.00E+8nM ΔG°: >-0.564kcal/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair