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TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433865(CHEMBL2380402)
Affinity DataKi:  4nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataKi:  5nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433878(CHEMBL2380389)
Affinity DataKi:  6nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433880(CHEMBL2380387)
Affinity DataKi:  6.20nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataKi:  6.60nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433877(CHEMBL2380390)
Affinity DataKi:  7nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50592895(CHEMBL5187653)
Affinity DataKi:  10nMAssay Description:Inhibition of MMP-14 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433871(CHEMBL2380396)
Affinity DataKi:  10nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433868(CHEMBL2380400)
Affinity DataKi:  11nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50343077(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(trifluoromet...)
Affinity DataKi:  14nMAssay Description:Inhibition of human MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433866(CHEMBL2380314)
Affinity DataKi:  21nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078947((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-[2-[1-ca...)
Affinity DataKi:  22nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50423397(CHEMBL398271)
Affinity DataKi:  26nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078937((1-Benzyloxycarbonylamino-ethyl)-{3-benzylsulfanyl...)
Affinity DataKi:  26nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433872(CHEMBL2380395)
Affinity DataKi:  31nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433872(CHEMBL2380395)
Affinity DataKi:  31nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078935((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  32nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50264809(Thiirane, 1 | Thiirane (deuterium), 1-d2 | CHEMBL4...)
Affinity DataKi:  37nMAssay Description:Competitive inhibition of human MMP14 using fluorogenic substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM408486(US10357546, ND-3640)
Affinity DataKi:  40nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078951([1-(2-Benzyloxy-acetylamino)-2-phenyl-ethyl]-{2-[1...)
Affinity DataKi:  40nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078950((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  41nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078946([1-(2-Benzyloxycarbonylamino-propionylamino)-2-phe...)
Affinity DataKi:  41nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078945((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  45nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50104710(2-Benzenesulfonylamino-N-[5-(4-chloro-phenyl)-6H-[...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloprotease-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078941([1-(2-Benzyloxycarbonylamino-4-methyl-pentanoylami...)
Affinity DataKi:  53nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50459506(CHEMBL4214929)
Affinity DataKi:  53nMAssay Description:Slow binding inhibition of human recombinant MMP14 catalytic domain using MOCAc-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078932((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  60nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataKi:  62nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataKi:  62nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078929((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  63nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433875(CHEMBL2380392)
Affinity DataKi:  68nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50616392(CHEMBL5412341)
Affinity DataKi:  68nMAssay Description:Inhibition of human recombinant MMP14 using MOCAc-Lys-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-N2 as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50265157((6S,7S)-N-hydroxy-5-methyl-6-(4-(5-(trifluoromethy...)
Affinity DataKi:  68nMAssay Description:Inhibition of recombinant human MMP14 catalytic domain (89 to 265 residues) expressed in Escherichia coli using MOCAc-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50433879(CHEMBL2380388)
Affinity DataKi:  70nMAssay Description:Inhibition of MMP-14 (unknown origin) using Mca-PLGLDpa-AR-NH2 as substrate preincubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078928((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  73nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50388914(CHEMBL2063274 | US10357546, p-OH SB-3CT)
Affinity DataKi:  90nMAssay Description:Competitive inhibition of human MMP14 using fluorogenic substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078943((1-Acetylamino-2-phenyl-ethyl)-{2-[1-carbamoyl-2-(...)
Affinity DataKi:  90nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50423403(CHEMBL251253)
Affinity DataKi:  91nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078954((1-Benzyloxycarbonylamino-ethyl)-{2-[1-carbamoyl-2...)
Affinity DataKi:  92nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50102594(7-Isobutyl-8-oxo-2-oxa-9-aza-bicyclo[10.2.2]hexade...)
Affinity DataKi:  94nMAssay Description:Inhibition of matrix metalloprotease-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50104721((S)-N-(5-(4-chlorophenyl)-6H-1,3,4-thiadiazin-2-yl...)
Affinity DataKi:  100nMAssay Description:In vitro inhibitory activity against the catalytic domain of human matrix metalloprotease-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50354624(CHEMBL1834422 | US9951035, ND-322 (2) | US10357546...)
Affinity DataKi:  100nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM92441(RXP470, Compound 4 | RXP470, 1)
Affinity DataKi: >100nM ΔG°: >-9.54kcal/molepH: 6.8 T: 2°CAssay Description:Enzyme assay using human matrix metalloproteases or ADAMTS.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50138684((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  105nMAssay Description:Inhibition of Matrix metalloprotease-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50138684((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  105nMAssay Description:Binding affinity to MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50078930((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[(R)-...)
Affinity DataKi:  105nMAssay Description:Binding affinity against matrix metalloprotease-14 MTI-MMP.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50393211(CHEMBL2153737)
Affinity DataKi:  105nMAssay Description:Inhibition of MMP-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50104723(2-Benzenesulfonylamino-N-[5-(4-chloro-phenyl)-6H-[...)
Affinity DataKi:  110nMAssay Description:In vitro inhibitory activity against the ectodomain of the human matrix metalloproteinase-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50264809(Thiirane, 1 | Thiirane (deuterium), 1-d2 | CHEMBL4...)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant MMP14 catalytic domain by substrate hydrolysis based fluorescence spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Florida State University

Curated by ChEMBL
LigandPNGBDBM50264809(Thiirane, 1 | Thiirane (deuterium), 1-d2 | CHEMBL4...)
Affinity DataKi:  110nMAssay Description:Inhibition of MMP-14 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
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