TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 520nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 760nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataKi: 7.90E+3nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate measured for 120 min...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of immunoproteasome-20S subunit beta5i in human PBMC assessed as substrate hydrolysis using suc-LLVY-AMC as substrate preincubated for 15 ...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataEC50: 4.20E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Weill Cornell Medical College
Curated by ChEMBL
Weill Cornell Medical College
Curated by ChEMBL
Affinity DataEC50: 1.54E+4nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...More data for this Ligand-Target Pair