Affinity DataKi: 0.5nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 136nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 870nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.33E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+4nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
Affinity DataEC50: 0.210nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 0.0230nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor delta 1 in functional assa...More data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay,G...More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+4nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay,G...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 0.0550nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 7.30E+3nMAssay Description:In vitro bioassay data to determine the effective concentration required for antagonistic activity against Opioid receptor mu 1 in functional assay,G...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 0.0360nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0570nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.670nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.130nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataEC50: 0.0910nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair