Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50040098
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389160(CHEMBL2064741)
Affinity DataEC50:  325nMAssay Description:Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389161(CHEMBL2064742)
Affinity DataEC50:  682nMAssay Description:Agonist activity at PPARgamma LBD in human 293H DA cells after 16 hrs by TR-FRET activation reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389162(CHEMBL2064743)
Affinity DataEC50:  2.40E+3nMAssay Description:Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  190nMAssay Description:Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataEC50:  26nMAssay Description:Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389160(CHEMBL2064741)
Affinity DataEC50:  215nMAssay Description:Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389161(CHEMBL2064742)
Affinity DataEC50:  5.45E+3nMAssay Description:Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389162(CHEMBL2064743)
Affinity DataEC50:  2.40E+3nMAssay Description:Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  120nMAssay Description:Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataEC50:  3.70nMAssay Description:Displacement of pan-PPAR fluormone from PPARgamma LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389160(CHEMBL2064741)
Affinity DataEC50:  467nMAssay Description:Agonist activity at PPARgamma LBD in human 293H DA cells after 16 hrs by TR-FRET activation reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389162(CHEMBL2064743)
Affinity DataEC50:  594nMAssay Description:Agonist activity at PPARgamma LBD in human 293H DA cells after 16 hrs by TR-FRET activation reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at PPARgamma LBD in human 293H DA cells after 16 hrs by TR-FRET activation reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389161(CHEMBL2064742)
Affinity DataEC50:  1.14E+4nMAssay Description:Displacement of pan-PPAR fluormone from PPARalpha LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataEC50:  5.53E+4nMAssay Description:Displacement of pan-PPAR fluormone from PPARalpha LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  1.80nMAssay Description:Displacement of pan-PPAR fluormone from PPARalpha LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  920nMAssay Description:Displacement of pan-PPAR fluormone from PPARalpha LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389161(CHEMBL2064742)
Affinity DataEC50:  2.10E+4nMAssay Description:Displacement of pan-PPAR fluormone from PPARdelta LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389162(CHEMBL2064743)
Affinity DataEC50:  2.60E+4nMAssay Description:Displacement of pan-PPAR fluormone from PPARdelta LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  2.90nMAssay Description:Displacement of pan-PPAR fluormone from PPARdelta LBD by TR-FRET based LanthaScreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50389161(CHEMBL2064742)
Affinity DataEC50:  5.45E+3nMAssay Description:Binding affinity to PPARgamma LBD by fluorescence polarization based competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed