TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at mGluR5 in mouse astrocytes assessed as inhibition of L-quisqualate induced calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at mGluR5 in mouse astrocytes assessed as inhibition of L-quisqualate induced calcium release by FLIPR assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 5.01E+3nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: <3.16E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: <3.16E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: <3.16E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: 3.16E+4nMAssay Description:Antagonist activity at mGluR5More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: <3.16E+4nMAssay Description:Antagonist activity at human mGluR5 expressed in CHO cells assessed as doxycycline induced calcium mobilizationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Medicines Research Centre
Curated by ChEMBL
Medicines Research Centre
Curated by ChEMBL
Affinity DataIC50: <5.01E+4nMAssay Description:Antagonist activity at mGluR5More data for this Ligand-Target Pair