Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50004746
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  0.765nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485612(GOMISIN A)
Affinity DataIC50:  0.960nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485610(SCHIZANDRIN | Schisandrin)
Affinity DataIC50:  1.16nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50341711(CHEMBL479488 | schisandrin B)
Affinity DataIC50:  1.25nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  6.32nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485611(SCHISANDRIN A)
Affinity DataIC50:  6.96nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485610(SCHIZANDRIN | Schisandrin)
Affinity DataIC50:  8.09nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485612(GOMISIN A)
Affinity DataIC50:  9.36nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50341711(CHEMBL479488 | schisandrin B)
Affinity DataIC50:  9.49nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485611(SCHISANDRIN A)
Affinity DataIC50:  9.84nMAssay Description:TP_TRANSPORTER: inhibition of VCR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  110nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485612(GOMISIN A)
Affinity DataIC50:  122nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485610(SCHIZANDRIN | Schisandrin)
Affinity DataIC50:  124nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50341711(CHEMBL479488 | schisandrin B)
Affinity DataIC50:  139nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485611(SCHISANDRIN A)
Affinity DataIC50:  141nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485611(SCHISANDRIN A)
Affinity DataIC50:  153nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  162nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485612(GOMISIN A)
Affinity DataIC50:  182nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50341711(CHEMBL479488 | schisandrin B)
Affinity DataIC50:  204nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485610(SCHIZANDRIN | Schisandrin)
Affinity DataIC50:  217nMAssay Description:TP_TRANSPORTER: inhibition of DNR transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  1.63E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50341711(CHEMBL479488 | schisandrin B)
Affinity DataIC50:  2.24E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485611(SCHISANDRIN A)
Affinity DataIC50:  2.33E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485612(GOMISIN A)
Affinity DataIC50:  2.76E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485609(SCHISANTHERIN A)
Affinity DataIC50:  3.05E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485610(SCHIZANDRIN | Schisandrin)
Affinity DataIC50:  3.23E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/MRP cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50341711(CHEMBL479488 | schisandrin B)
Affinity DataIC50:  4.18E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485611(SCHISANDRIN A)
Affinity DataIC50:  4.88E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485610(SCHIZANDRIN | Schisandrin)
Affinity DataIC50:  7.24E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50485612(GOMISIN A)
Affinity DataIC50:  7.77E+3nMAssay Description:TP_TRANSPORTER: inhibition of VP-16 transport in HL60/ADR cells (overexpression of MRP1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed