Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50006327
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498871(CHEMBL97313)
Affinity DataKi:  43nMAssay Description:Competitive inhibition of Escherichia coli DHFR by Lineweaver-Burk plot analysis in presence of H2FMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498871(CHEMBL97313)
Affinity DataKi:  50nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498878(CHEMBL97567)
Affinity DataKi:  93nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498878(CHEMBL97567)
Affinity DataKi:  101nMAssay Description:Competitive inhibition of Escherichia coli DHFR by Lineweaver-Burk plot analysis in presence of H2FMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498873(CHEMBL94742)
Affinity DataKi:  359nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498873(CHEMBL94742)
Affinity DataKi:  394nMAssay Description:Competitive inhibition of Escherichia coli DHFR by Lineweaver-Burk plot analysis in presence of H2FMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498874(CHEMBL1617293)
Affinity DataKi:  430nMAssay Description:Competitive inhibition of Escherichia coli DHFR by Lineweaver-Burk plot analysis in presence of H2FMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498874(CHEMBL1617293)
Affinity DataKi:  880nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50291779(3-(4,6-Diamino-2,2-dimethyl-2H-[1,3,5]triazin-1-yl...)
Affinity DataKi:  958nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM18792(1-(4-chlorophenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-...)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50090051(6,6-Dimethyl-1-p-tolyl-1,6-dihydro-[1,3,5]triazine...)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498877(CHEMBL316611)
Affinity DataKi:  2.89E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498877(CHEMBL316611)
Affinity DataKi:  3.82E+3nMAssay Description:Competitive inhibition of Escherichia coli DHFR by Lineweaver-Burk plot analysis in presence of H2FMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50405035(CHEMBL266573)
Affinity DataKi:  4.02E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498872(CHEMBL333873)
Affinity DataKi:  1.12E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50031299(6-(2,3-Dichloro-phenyl)-[1,2,4]triazine-3,5-diamin...)
Affinity DataKi:  1.52E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498880(CHEMBL1625056)
Affinity DataKi:  2.02E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498876(CHEMBL3634634)
Affinity DataKi:  3.93E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498879(CHEMBL1412044)
Affinity DataKi:  1.05E+5nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formation by quadratic Morrison plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498871(CHEMBL97313)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498878(CHEMBL97567)
Affinity DataIC50:  1.84E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498873(CHEMBL94742)
Affinity DataIC50:  7.59E+3nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498874(CHEMBL1617293)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50291779(3-(4,6-Diamino-2,2-dimethyl-2H-[1,3,5]triazin-1-yl...)
Affinity DataIC50:  2.02E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM18792(1-(4-chlorophenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-...)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50090051(6,6-Dimethyl-1-p-tolyl-1,6-dihydro-[1,3,5]triazine...)
Affinity DataIC50:  3.23E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498877(CHEMBL316611)
Affinity DataIC50:  6.28E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50405035(CHEMBL266573)
Affinity DataIC50:  8.91E+4nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498872(CHEMBL333873)
Affinity DataIC50:  2.63E+5nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50031299(6-(2,3-Dichloro-phenyl)-[1,2,4]triazine-3,5-diamin...)
Affinity DataIC50:  3.49E+5nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498880(CHEMBL1625056)
Affinity DataIC50:  4.78E+5nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498876(CHEMBL3634634)
Affinity DataIC50:  7.22E+5nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498879(CHEMBL1412044)
Affinity DataIC50:  1.55E+6nMAssay Description:Inhibition of Escherichia coli DHFR assessed as NADP formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498880(CHEMBL1625056)
Affinity DataKd:  3.32E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498873(CHEMBL94742)
Affinity DataKd:  340nMAssay Description:Binding affinity to Escherichia coli DHFR at 10 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498875(CHEMBL97830)
Affinity DataKd:  8.26E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM18792(1-(4-chlorophenyl)-6,6-dimethyl-1,6-dihydro-1,3,5-...)
Affinity DataKd:  1.18E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50405035(CHEMBL266573)
Affinity DataKd:  1.72E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498874(CHEMBL1617293)
Affinity DataKd:  6.16E+3nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50090051(6,6-Dimethyl-1-p-tolyl-1,6-dihydro-[1,3,5]triazine...)
Affinity DataKd:  9.32E+3nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498881(CHEMBL589682 | SJ000034418)
Affinity DataKd:  1.85E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498876(CHEMBL3634634)
Affinity DataKd:  1.45E+5nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498872(CHEMBL333873)
Affinity DataKd:  2.45E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498878(CHEMBL97567)
Affinity DataKd:  10nMAssay Description:Binding affinity to Escherichia coli DHFR at 10 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498877(CHEMBL316611)
Affinity DataKd:  730nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498879(CHEMBL1412044)
Affinity DataKd:  4.80E+4nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50498871(CHEMBL97313)
Affinity DataKd:  6.93E+3nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Escherichia coli)
Georgia Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50291779(3-(4,6-Diamino-2,2-dimethyl-2H-[1,3,5]triazin-1-yl...)
Affinity DataKd:  8.74E+3nMAssay Description:Binding affinity to Escherichia coli DHFR at 500 uM using spyro orange reporter dye by differential scanning fluorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed