Compile Data Set for Download or QSAR
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Found 38 Enz. Inhib. hit(s) with all data for entry = 50015932
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM21190(4-(2-{[5-amino-2-(furan-2-yl)-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50394715(CHEMBL2165804)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50382491(CHEMBL2024114 | US10988455, Example 1(xlii))
Affinity DataKi:  4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590625(CHEMBL5206530)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590626(CHEMBL5199840)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590616(CHEMBL5206491)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590619(CHEMBL5188677)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590621(CHEMBL5196511)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590617(CHEMBL5169415)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50548112(CHEMBL4791612)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590618(CHEMBL5200008)
Affinity DataKi:  456nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590610(CHEMBL5179562)
Affinity DataKi:  586nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590613(CHEMBL5198386)
Affinity DataKi:  651nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590620(CHEMBL5178327)
Affinity DataKi:  696nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590612(CHEMBL5172270)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590611(CHEMBL5208266)
Affinity DataKi:  736nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590607(CHEMBL5192778)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590615(CHEMBL5185932)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50354815(CHEMBL1834385)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590600(CHEMBL2357789)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590608(CHEMBL5183274)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590599(CHEMBL5179156)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590603(CHEMBL5183517)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590602(CHEMBL5174569)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590601(CHEMBL5186870)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590605(CHEMBL1729531)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM3255(4-Anilino quinazoline deriv. 6 | N-(2-phenylethyl)...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590622(CHEMBL25099)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50177832(CHEMBL3815078)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50177805(CHEMBL3814123)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590623(CHEMBL4587670)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590624(CHEMBL1588916)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590609(CHEMBL5183199)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590606(CHEMBL5196537)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590614(CHEMBL5183860)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50590604(CHEMBL5175024)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed