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Found 140 Enz. Inhib. hit(s) with all data for entry = 50018771
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50323167((5-(2,4-dichlorophenyl)-2-(4-methoxyphenyl)-7-meth...)
Affinity DataKi:  5.60E+3nMAssay Description:Binding affinity to DPP-4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50323161((5-(2,4-dichlorophenyl)-7-methyl-2-phenylimidazo[1...)
Affinity DataKi:  6.00E+3nMAssay Description:Binding affinity to DPP-4 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50323187(6-(aminomethyl)-7-(2,4-dichlorophenyl)-N-(2-methox...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of DPP-8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612351(CHEMBL5269774)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of DPP-9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612351(CHEMBL5269774)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of DPP-8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612350(CHEMBL5275567)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of DPP-8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612350(CHEMBL5275567)
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of DPP-9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612314(CHEMBL5279548)
Affinity DataIC50:  0.0270nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50135009(CHEMBL3736423)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612333(CHEMBL5267753)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612327(CHEMBL5279910)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612328(CHEMBL5268418)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612329(CHEMBL5273218)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612330(CHEMBL5275162)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612331(CHEMBL5277064)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612332(CHEMBL3736190)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM107101(US8592371, 3)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612334(CHEMBL5283277)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612335(CHEMBL5276887)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612336(CHEMBL3735329)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612337(CHEMBL3736085)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM222244(6-Iodo-N3-(3-nitrobenzylidene)-2-phenyl-N4-(thiazo...)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of DPP-4 (unknown origin) using (H-Gly-Pro-AMC) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612363(CHEMBL5279474)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612352(CHEMBL5274129)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612354(CHEMBL5276657)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612355(CHEMBL5265910)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612356(CHEMBL5269746)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612357(CHEMBL5277828)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612358(CHEMBL5269884)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612359(CHEMBL5273793)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612361(CHEMBL5276298)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612362(CHEMBL5289339)
Affinity DataIC50:  0.870nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612353(CHEMBL5272644)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612360(CHEMBL5275046)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612346(CHEMBL5276961)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612373(CHEMBL5288974)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP-4 (unknown origin) using (H-Gly-Pro-AMC) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human recombinant DPP-4 using (H-Gly-Pro-AMC as substrateMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612342(CHEMBL5277490)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612371(CHEMBL5279728)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human recombinant DPP-4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50612314(CHEMBL5279548)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of DPP-9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50516918(CHEMBL4446618)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of human recombinant DPP-4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50257317((S)-1-((S)-2-amino-5-(isoindolin-2-yl)-5-oxopentan...)
Affinity DataIC50:  2nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612345(CHEMBL5271401)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50420657(CHEMBL2086613)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human recombinant DPP-4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50612314(CHEMBL5279548)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of DPP-8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of human recombinant DPP-4More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50612297(CHEMBL5267474)
Affinity DataIC50:  3nMAssay Description:Inhibition of DPP-4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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