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Found 4 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 50012609
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50558736(CHEMBL4756472)
Affinity DataEC50:  68nMAssay Description:Irreversible agonist activity at human adenosine A2A receptor expressed in Flp-In-CHO cells assessed as effect on forskolin-induced cAMP accumulation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataEC50:  2.5nMAssay Description:Irreversible agonist activity at human adenosine A2A receptor expressed in Flp-In-CHO cells assessed as effect on forskolin-induced cAMP accumulation...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50558738(CHEMBL4746617)
Affinity DataEC50:  68nMAssay Description:Irreversible agonist activity at human adenosine A2A receptor expressed in Flp-In-CHO cells assessed as effect on forskolin-induced cAMP accumulation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50558737(CHEMBL4741079)
Affinity DataEC50:  646nMAssay Description:Irreversible agonist activity at human adenosine A2A receptor expressed in Flp-In-CHO cells assessed as effect on forskolin-induced cAMP accumulation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed