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Found 6 of ec50 data for polymerid = 7230
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Shaanxi Province Tuberculosis Prevention And Treatment Institute

Curated by ChEMBL
LigandPNGBDBM50503709(CHEMBL4588123)
Affinity DataEC50:  420nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Shaanxi Province Tuberculosis Prevention And Treatment Institute

Curated by ChEMBL
LigandPNGBDBM50503710(CHEMBL4475584)
Affinity DataEC50:  500nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Shaanxi Province Tuberculosis Prevention And Treatment Institute

Curated by ChEMBL
LigandPNGBDBM50503708(CHEMBL4457385)
Affinity DataEC50:  1.99E+3nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Shaanxi Province Tuberculosis Prevention And Treatment Institute

Curated by ChEMBL
LigandPNGBDBM50503711(CHEMBL4447072)
Affinity DataEC50:  4.64E+3nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Shaanxi Province Tuberculosis Prevention And Treatment Institute

Curated by ChEMBL
LigandPNGBDBM50525863(CHEMBL1708524)
Affinity DataEC50:  1.17E+4nMAssay Description:Inhibition of PDK1 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Shaanxi Province Tuberculosis Prevention And Treatment Institute

Curated by ChEMBL
LigandPNGBDBM50177027(CPC-211 | Ceresine | DCA | Sodium dichloroacetate)
Affinity DataEC50:  5.70E+6nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed