Compile Data Set for Download or QSAR
Report error Found 286 Enz. Inhib. hit(s) with all data for entry = 744
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289071BDBM289071(US10093640, Example 279 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289072BDBM289072(US10093640, Example 299 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289075BDBM289075(US10093640, Example 300 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289076BDBM289076(US10093640, Example 301 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289078BDBM289078(US10093640, Example 302 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289079BDBM289079(US10093640, Example 303 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289080BDBM289080(US10093640, Example 304 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50160010BDBM50160010(CHEMBL3786147 | US10093640, Example 305 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289022BDBM289022(US10093640, Example 233 | 6-chloro-3-(3-(4-chloro-...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50159954BDBM50159954(CHEMBL3785998 | US10093640, Example 237 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50159945BDBM50159945(CHEMBL3785666 | US10093640, Example 253 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50159940BDBM50159940(CHEMBL3785228 | US10093640, Example 255 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289051BDBM289051(US10093640, Example 260 | -chloro-3-(3-(4-chloro-3...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289052BDBM289052(US10093640, Example 261 | 5-(N-(6-chloro-3-(3-(4-c...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289055BDBM289055(US10093640, Example 264 | methyl 5-(N-(6-chloro-3-...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289058BDBM289058(US10093640, Example 266 | 5-(N-(6-chloro-3-(3-(4-c...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289082BDBM289082(US10093640, Example 306 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289083BDBM289083(US10093640, Example 307 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289084BDBM289084(US10093640, Example 308 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38104BDBM38104(US10093640, Example 92 | 3-(3-(4-chloro-3,5-dimeth...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38109BDBM38109(US10093640, Example 98 | 3-(3-(4-chloro-3,5-dimeth...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38110BDBM38110(US10093640, Example 99 | 3-(3-(4-chloro-3,5-dimeth...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38112BDBM38112(US10093640, Example 100 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38114BDBM38114(US10093640, Example 101 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38115BDBM38115(US10093640, Example 102 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38119BDBM38119(US10093640, Example 103 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38120BDBM38120(US10093640, Example 104 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38065BDBM38065(US10093640, Example 50 | 4-chloro-3-(3-(4-chloro-3...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38066BDBM38066(US10093640, Example 51 | 4-chloro-3-(3-(4-chloro-3...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38101BDBM38101(US10093640, Example 88 | 3-(3-(4-chloro-3,5-dimeth...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50160000BDBM50160000(CHEMBL3786018 | US10093640, Example 89 | US1084403...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38103BDBM38103(US10093640, Example 90 | 3-(3-(4-chloro-3,5-dimeth...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 286515BDBM286515(US10093640, Example 204 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 286516BDBM286516(US10093640, Example 205 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 286517BDBM286517(US10093640, Example 206 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 286518BDBM286518(US10093640, Example 207 | N-((2-(1-benzyl-1H-pyrro...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50159949BDBM50159949(CHEMBL3787178 | US10093640, Example 216 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50160018BDBM50160018(CHEMBL3785155 | US10093640, Example 226 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 289018BDBM289018(US10093640, Example 230 | 6-chloro-3-(3-(4-chloro-...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50159933BDBM50159933(CHEMBL3786092 | US10093640, Example 232 | US108440...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38131BDBM38131(US10093640, Example 113 | 4-bromo-3-(3-(4-chloro-3...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38134BDBM38134(US10093640, Example 116 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38141BDBM38141(US10093640, Example 121 | 6-chloro-3-(3-(4-chloro-...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38143BDBM38143(US10093640, Example 123 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38144BDBM38144(US10093640, Example 124 | 7-(3-((4-(4-acetylpipera...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38147BDBM38147(US10093640, Example 127 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38150BDBM38150(US10093640, Example 130 | 3-(3-(4-chloro-3,5-dimet...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 38201BDBM38201(US10093640, Example 170 | 33-(3-(4-chloro-3,5-dime...)
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50424725BDBM50424725(CHEMBL2314177 | US10093640, Example 5 | US10844032...)
Affinity DataIC50: 120nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 50424725BDBM50424725(CHEMBL2314177 | US10093640, Example 5 | US10844032...)
Affinity DataIC50: 200nMpH: 7.5 T: 2°CAssay Description:Compound affinity was measured using a fluorescence polarization anisotropy competition assay. Anisotropy measurements were carried out in 384-well, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

Displayed 1 to 50 (of 286 total ) | Next | Last >>
Jump to: