Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 11692
TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640362BDBM640362(3-((8-amino-3-isopropylimidazo[1,5-a]pyrazin-1-yl)...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640363BDBM640363(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640363BDBM640363(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640364BDBM640364(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640361BDBM640361(3-((8-amino-3-methylimidazo[1,5-a]pyrazin-1-yl)eth...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640361BDBM640361(3-((8-amino-3-methylimidazo[1,5-a]pyrazin-1-yl)eth...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640362BDBM640362(3-((8-amino-3-isopropylimidazo[1,5-a]pyrazin-1-yl)...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640366BDBM640366(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640367BDBM640367(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640367BDBM640367(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640364BDBM640364(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640365BDBM640365(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640366BDBM640366(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640359BDBM640359(3-((8-amino-3-ethylimidazo[1,5-a]pyrazin-1-yl)ethy...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640359BDBM640359(3-((8-amino-3-ethylimidazo[1,5-a]pyrazin-1-yl)ethy...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640379BDBM640379(N-(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640380BDBM640380(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-pyr...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640376BDBM640376(N-(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640377BDBM640377(N-(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640377BDBM640377(N-(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640383BDBM640383(N-(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640383BDBM640383(N-(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640380BDBM640380(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-pyr...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640381BDBM640381(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-pyr...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640382BDBM640382(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-pyr...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640372BDBM640372(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640369BDBM640369(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640374BDBM640374(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640375BDBM640375(N-(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640375BDBM640375(N-(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640376BDBM640376(N-(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640372BDBM640372(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640373BDBM640373(3-((4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640373BDBM640373(3-((4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640374BDBM640374(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-...)
Affinity DataIC50: 5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640379BDBM640379(N-(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640378BDBM640378(N-(3-((4-amino-7-cyclopentyl-7H-pyrrolo[2,3-d]pyri...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640382BDBM640382(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-pyr...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640368BDBM640368(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640365BDBM640365(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640381BDBM640381(3-((4-amino-7-((1r,4r)-4-hydroxycyclohexyl)-7H-pyr...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640370BDBM640370(3-((4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640371BDBM640371(3-((4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640371BDBM640371(3-((4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640368BDBM640368(3-((4-amino-7-ethyl-7H-pyrrolo[2,3-d]pyrimidin-5-y...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640369BDBM640369(3-((4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640370BDBM640370(3-((4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidin...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640360BDBM640360(3-((8-amino-3-ethylimidazo[1,5-a]pyrazin-1-yl)ethy...)
Affinity DataIC50: 27.5nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640378BDBM640378(N-(3-((4-amino-7-cyclopentyl-7H-pyrrolo[2,3-d]pyri...)
Affinity DataIC50: 75nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Shenzhen Targetrx

US Patent
LigandChemical structure of BindingDB Monomer ID 640360BDBM640360(3-((8-amino-3-ethylimidazo[1,5-a]pyrazin-1-yl)ethy...)
Affinity DataIC50: 75nMAssay Description:Specific Assay Method:Compound formulation: The test compounds were dissolved in DMSO to prepare a 20 mM stock solution. Before use, the compounds we...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2024
Entry Details
US Patent