Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50040201
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Tennessee Medical Center

Curated by ChEMBL
LigandPNGBDBM50390978(VALSPODAR)
Affinity DataKi:  1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of Calcein-AM efflux in CEM/VBL 100 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Tennessee Medical Center

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  1.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Calcein-AM efflux in CEM/VLB100 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
University Of Tennessee Medical Center

Curated by ChEMBL
LigandPNGBDBM50423876(DEXNIGULDIPINE)
Affinity DataKi:  2.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of Calcein-AM efflux in CEM/VLB100 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed