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Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50036768
TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082611(3,3-Dimethyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  5.70nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082575(3,3-Dimethyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  6nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082578(6-Chloro-3,3-dimethyl-1,2,3,4-tetrahydro-quinoline...)
Affinity DataKi:  6.60nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082589(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  11nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082579(6-Chloro-3,3-dimethyl-1,2,3,4-tetrahydro-quinoline...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082583(Acetic acid 2-{1-[5-guanidino-2-(3-methyl-1,2,3,4-...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082589(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082598(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  23nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082577(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  23nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082612(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082580(3,3-Dimethyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  32nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082608(CHEMBL139718 | Succinic acid mono-(2-{1-[5-guanidi...)
Affinity DataKi:  34nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082581(CHEMBL143203 | N-(2-{1-[2-(3,3-Dimethyl-1,2,3,4-te...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082573(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  44nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082591(CHEMBL139606 | N-(2-{1-[5-Guanidino-2-(3-methyl-1,...)
Affinity DataKi:  45nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082603((R)-3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  46nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082580(3,3-Dimethyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082594(CHEMBL356067 | N-[1-(3,4-Dihydro-1H-isoquinoline-2...)
Affinity DataKi:  49nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082573(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  52nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082597(2,2-Dimethyl-propionic acid 2-{1-[2-(6-chloro-3,3-...)
Affinity DataKi:  56nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataKi:  61nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataKi:  61nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082610(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  64nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082602(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  64nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082591(CHEMBL139606 | N-(2-{1-[5-Guanidino-2-(3-methyl-1,...)
Affinity DataKi:  66nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082592(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082595(CHEMBL140469 | N-[4-Guanidino-1-(pyrrolidine-1-car...)
Affinity DataKi:  110nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082572(CHEMBL337532 | Pentanedioic acid mono-(2-{1-[5-gua...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082587(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  185nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082606(3-(3-{1-[5-Guanidino-2-(3-methyl-1,2,3,4-tetrahydr...)
Affinity DataKi:  280nMAssay Description:The compound was evaluated for the inhibitory activity against human thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082606(3-(3-{1-[5-Guanidino-2-(3-methyl-1,2,3,4-tetrahydr...)
Affinity DataKi:  310nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082584(CHEMBL435785 | Malonic acid mono-(2-{1-[5-guanidin...)
Affinity DataKi:  360nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082605(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  360nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082600(1,2,3,4-Tetrahydro-quinoline-8-sulfonic acid {4-gu...)
Affinity DataKi:  490nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082604(CHEMBL140686 | N-(2-{1-[5-Guanidino-2-(3-methyl-1,...)
Affinity DataKi:  650nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082574(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  795nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082596(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  890nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082607(4-(2-{1-[5-Guanidino-2-(3-methyl-1,2,3,4-tetrahydr...)
Affinity DataKi:  980nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082590((2S,4S)-1-{5-Guanidino-2-[3-(1-methyl-1-phenyl-eth...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082571(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082576(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082599(7-{1-[5-Guanidino-2-(3-methyl-1,2,3,4-tetrahydro-q...)
Affinity DataKi:  1.98E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082586(CHEMBL143412 | {1-[5-Guanidino-2-(3-methyl-1,2,3,4...)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082609(CHEMBL140911 | N-[4-Guanidino-1-((S)-2-hydroxymeth...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082601(CHEMBL143226 | N-[4-Guanidino-1-((S)-2-hydroxymeth...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082585(3-Methyl-1,2,3,4-tetrahydro-quinoline-8-sulfonic a...)
Affinity DataKi:  5.18E+3nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAnionic trypsin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082580(3,3-Dimethyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  7.10E+3nMAssay Description:The compound was evaluated for the inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082593(3-{1-[5-Guanidino-2-(3-methyl-1,2,3,4-tetrahydro-q...)
Affinity DataKi:  1.84E+4nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082582(CHEMBL262213 | [2-(2-{1-[5-Guanidino-2-(3-methyl-1...)
Affinity DataKi:  3.52E+4nMAssay Description:Inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetChymotrypsinogen A(Bovine)
Novartis Horsham Research Centre

Curated by ChEMBL
LigandPNGBDBM50082580(3,3-Dimethyl-1,2,3,4-tetrahydro-quinoline-8-sulfon...)
Affinity DataKi:  8.30E+4nMAssay Description:The compound was evaluated for the inhibitory activity against bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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