Found 39 Enz. Inhib. hit(s) with all data for entry = 50003574 
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibitory constant determined using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibitory constant against human Alpha-2A adrenergic receptor expressed in LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 102nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Inhibitory constant, using [3H]rauwolscine in LM(tk-) cells stably transfected with cloned human Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Inhibitory constant against human Alpha-2B adrenergic receptor expressed in Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Alpha-2A adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Alpha-2C adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Alpha-2A adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Alpha-2A adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Alpha-2B adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 71nMAssay Description:Alpha-2A adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 9.30nMAssay Description:Alpha-2B adrenergic receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Alpha2c receptor agonism measured as ability to inhibit forskolin-stimulated synthesis of cAMPMore data for this Ligand-Target Pair
