Compile Data Set for Download or QSAR
Report error Found 236 Enz. Inhib. hit(s) with all data for entry = 50010312
TargetTryptase gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093142BDBM50093142(APC-1390 | 1N-(3,3-diphenylpropyl)-4-[4-amino(imin...)
Affinity DataKd:  0.0700nMAssay Description:Dissociation constant of compound was evaluated from its IC50 against tryptase at different concentrationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093175BDBM50093175(Derivative of APC-2059 | CHEMBL311655)
Affinity DataKi:  0.100nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093157BDBM50093157(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  0.100nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093153BDBM50093153(Derivative of APC-2059 | CHEMBL306620)
Affinity DataKd:  0.100nMAssay Description:Dissociation constant of compound was evaluated from its IC50 against tryptase at different concentrationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093192BDBM50093192(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  0.200nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093167BDBM50093167(Derivative of APC-2059 | CHEMBL75750)
Affinity DataKi:  0.400nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093156BDBM50093156(Derivative of APC-2059 | CHEMBL432172)
Affinity DataKi:  0.400nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093154BDBM50093154(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  0.400nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093199BDBM50093199(Derivative of APC-2059 | CHEMBL75972)
Affinity DataKi:  0.5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093173BDBM50093173(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  0.5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093158BDBM50093158(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  0.5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093178BDBM50093178(Derivative of APC-2059 | CHEMBL76883)
Affinity DataKi:  0.700nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093176BDBM50093176(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  1nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093197BDBM50093197(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  2nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093186BDBM50093186(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  2nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093198BDBM50093198(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093164BDBM50093164(Derivative of APC-2059 | CHEMBL308632)
Affinity DataKi:  3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093161BDBM50093161(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  4nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093148BDBM50093148(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  4nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093183BDBM50093183(Derivative of APC-2059 | CHEMBL76796)
Affinity DataKi:  4nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093168BDBM50093168(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093182BDBM50093182(Derivative of APC-2059 | CHEMBL77007)
Affinity DataKi:  8nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093187BDBM50093187(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  9nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093196BDBM50093196(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  10nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093190BDBM50093190(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  11nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093160BDBM50093160(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  16nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093184BDBM50093184(Derivative of APC-2059 | CHEMBL308074)
Affinity DataKi:  28nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093181BDBM50093181(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  30nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093191BDBM50093191(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  30nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093202BDBM50093202(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  44nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093170BDBM50093170(Derivative of APC-2059 | CHEMBL307427)
Affinity DataKi:  44nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093188BDBM50093188(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  70nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093193BDBM50093193(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  78nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093163BDBM50093163(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  80nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093169BDBM50093169(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  97nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093171BDBM50093171(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  100nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093151BDBM50093151(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  115nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093177BDBM50093177(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  180nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093166BDBM50093166(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  210nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093194BDBM50093194(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  240nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093180BDBM50093180(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  300nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093185BDBM50093185(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  440nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093159BDBM50093159(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  510nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093162BDBM50093162(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  610nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093200BDBM50093200(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  680nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093152BDBM50093152(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  820nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093172BDBM50093172(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  900nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093195BDBM50093195(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093179BDBM50093179(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTryptase beta-2/delta/gamma(Human)
Axys Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093203BDBM50093203(Derivative of piperazine-1-carboxylic acid 5-(pipe...)
Affinity DataKi:  1.00E+3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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