Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 1039
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8255BDBM8255(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(3-nitro...)
Affinity DataIC50: 20nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8271BDBM8271(2-chloro-5-{[4-(3-nitrophenyl)-2,5-dioxo-2,5-dihyd...)
Affinity DataIC50: 26nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8268BDBM8268(2-chloro-5-{[4-(2-nitrophenyl)-2,5-dioxo-2,5-dihyd...)
Affinity DataIC50: 28nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8252BDBM8252(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(2-nitro...)
Affinity DataIC50: 52nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8253BDBM8253(3-(3-chlorophenyl)-4-[(3,5-dichloro-4-hydroxypheny...)
Affinity DataIC50: 58nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8247BDBM8247(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-nitrophen...)
Affinity DataIC50: 59nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8229BDBM8229(3-[(3-chlorophenyl)amino]-4-(3-nitrophenyl)-2,5-di...)
Affinity DataIC50: 70nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8258BDBM8258(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(4-nitro...)
Affinity DataIC50: 71nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8267BDBM8267(2-chloro-5-{[4-(2-chlorophenyl)-2,5-dioxo-2,5-dihy...)
Affinity DataIC50: 74nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8269BDBM8269(2-chloro-5-{[4-(3-chlorophenyl)-2,5-dioxo-2,5-dihy...)
Affinity DataIC50: 76nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8263BDBM8263(3-{[4-(3-nitrophenyl)-2,5-dioxo-2,5-dihydro-1H-pyr...)
Affinity DataIC50: 79nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8251BDBM8251(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(2-metho...)
Affinity DataIC50: 82nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8257BDBM8257(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(4-metho...)
Affinity DataIC50: 83nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8270BDBM8270(2-chloro-5-{[4-(3-methoxyphenyl)-2,5-dioxo-2,5-dih...)
Affinity DataIC50: 85nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8256BDBM8256(3-(4-chlorophenyl)-4-[(3,5-dichloro-4-hydroxypheny...)
Affinity DataIC50: 91nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8250BDBM8250(3-(2-chlorophenyl)-4-[(3,5-dichloro-4-hydroxypheny...)
Affinity DataIC50: 93nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8246BDBM8246(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(3-chlorophe...)
Affinity DataIC50: 94nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8227BDBM8227(3-[(3-chlorophenyl)amino]-4-(2-nitrophenyl)-2,5-di...)
Affinity DataIC50: 104nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8272BDBM8272(2-chloro-5-{[4-(4-chlorophenyl)-2,5-dioxo-2,5-dihy...)
Affinity DataIC50: 109nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8275BDBM8275(3-(2-methoxyphenyl)-4-{[4-(methylsulfanyl)phenyl]a...)
Affinity DataIC50: 110nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8226BDBM8226(3-[(3-chlorophenyl)amino]-4-(2-methoxyphenyl)-2,5-...)
Affinity DataIC50: 114nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8241BDBM8241(3-[(4-hydroxyphenyl)amino]-4-(3-nitrophenyl)-2,5-d...)
Affinity DataIC50: 123nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8261BDBM8261(3-{[4-(3-chlorophenyl)-2,5-dioxo-2,5-dihydro-1H-py...)
Affinity DataIC50: 134nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8260BDBM8260(3-{[4-(2-chlorophenyl)-2,5-dioxo-2,5-dihydro-1H-py...)
Affinity DataIC50: 136nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8244BDBM8244(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(2-methoxyph...)
Affinity DataIC50: 139nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8221BDBM8221(3-(3-nitrophenyl)-4-(phenylamino)-2,5-dihydro-1H-p...)
Affinity DataIC50: 141nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8254BDBM8254(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-(3-metho...)
Affinity DataIC50: 142nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8266BDBM8266(2-chloro-5-[(2,5-dioxo-4-phenyl-2,5-dihydro-1H-pyr...)
Affinity DataIC50: 143nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8249BDBM8249(3-[(3,5-dichloro-4-hydroxyphenyl)amino]-4-phenyl-2...)
Affinity DataIC50: 149nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8243BDBM8243(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(2-chlorophe...)
Affinity DataIC50: 152nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8278BDBM8278(3-{[4-(methylsulfanyl)phenyl]amino}-4-(3-nitrophen...)
Affinity DataIC50: 152nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8231BDBM8231(3-[(3-chlorophenyl)amino]-4-(4-methoxyphenyl)-2,5-...)
Affinity DataIC50: 156nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8274BDBM8274(3-(2-chlorophenyl)-4-{[4-(methylsulfanyl)phenyl]am...)
Affinity DataIC50: 161nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8248BDBM8248(3-[(3-chloro-4-hydroxyphenyl)amino]-4-(4-chlorophe...)
Affinity DataIC50: 173nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8264BDBM8264(3-{[4-(4-chlorophenyl)-2,5-dioxo-2,5-dihydro-1H-py...)
Affinity DataIC50: 186nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8262BDBM8262(3-{[4-(3-methoxyphenyl)-2,5-dioxo-2,5-dihydro-1H-p...)
Affinity DataIC50: 195nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8225BDBM8225(3-(2-chlorophenyl)-4-[(3-chlorophenyl)amino]-2,5-d...)
Affinity DataIC50: 195nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8277BDBM8277(3-(3-methoxyphenyl)-4-{[4-(methylsulfanyl)phenyl]a...)
Affinity DataIC50: 203nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8265BDBM8265(3-{[4-(4-methoxyphenyl)-2,5-dioxo-2,5-dihydro-1H-p...)
Affinity DataIC50: 214nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8219BDBM8219(3-(2-chlorophenyl)-4-(phenylamino)-2,5-dihydro-1H-...)
Affinity DataIC50: 216nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8220BDBM8220(3-(2-methoxyphenyl)-4-(phenylamino)-2,5-dihydro-1H...)
Affinity DataIC50: 216nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8238BDBM8238(3-[(3-hydroxyphenyl)amino]-4-(3-nitrophenyl)-2,5-d...)
Affinity DataIC50: 236nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8280BDBM8280(3-(4-methoxyphenyl)-4-{[4-(methylsulfanyl)phenyl]a...)
Affinity DataIC50: 243nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8235BDBM8235(3-[(3-hydroxyphenyl)amino]-4-(2-nitrophenyl)-2,5-d...)
Affinity DataIC50: 251nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8228BDBM8228(3-[(3-chlorophenyl)amino]-4-(3-methoxyphenyl)-2,5-...)
Affinity DataIC50: 257nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8234BDBM8234(3-[(3-hydroxyphenyl)amino]-4-(2-methoxyphenyl)-2,5...)
Affinity DataIC50: 259nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8259BDBM8259(3-[(2,5-dioxo-4-phenyl-2,5-dihydro-1H-pyrrol-3-yl)...)
Affinity DataIC50: 291nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8224BDBM8224(3-[(3-chlorophenyl)amino]-4-phenyl-2,5-dihydro-1H-...)
Affinity DataIC50: 301nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8242BDBM8242(3-(4-chlorophenyl)-4-[(4-hydroxyphenyl)amino]-2,5-...)
Affinity DataIC50: 317nMAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Smithkline Beecham Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 8233BDBM8233(3-(2-chlorophenyl)-4-[(3-hydroxyphenyl)amino]-2,5-...)
Affinity DataIC50: 374nMpH: 7.0 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzyme and substrate in the presence 10 uM ATP/ [gamma-33P] ATP. Aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2006
Entry Details Article
PubMed
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