Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50010687
TargetSubstance-P receptor(Homo sapiens (Human))
Laboratoire De Chimie ThéRapeutique Associé

Curated by ChEMBL
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity towards Tachykinin receptor 1 expressed in CHO cells using [3H]-[Pro9]-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Laboratoire De Chimie ThéRapeutique Associé

Curated by ChEMBL
LigandPNGBDBM50097646((2-Methoxy-benzyl)-[1-(methylamino-phenyl-methyl)-...)
Affinity DataKi:  150nMAssay Description:Binding affinity towards Tachykinin receptor 1 expressed in CHO cells using [3H]-[Pro9]-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Laboratoire De Chimie ThéRapeutique Associé

Curated by ChEMBL
LigandPNGBDBM50097647((3,5-Bis-trifluoromethyl-benzyl)-[1-(methylamino-p...)
Affinity DataKi:  620nMAssay Description:Binding affinity towards Tachykinin receptor 1 expressed in CHO cells using [3H]-[Pro9]-SP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed