Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50037046
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116431({4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-yliden...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116424({4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-yliden...)
Affinity DataIC50: 7nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116419(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 11nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50: 11nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116424({4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-yliden...)
Affinity DataIC50: 38nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50334788((17beta-(N-tert-butylcarbamoyl)-4-aza-5alpha-andro...)
Affinity DataIC50: 41nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type I of human DU 145 prostatic tumor cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116429(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 60nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116418([4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ph...)
Affinity DataIC50: 75nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type 2 of human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116429(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 80nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116421(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116416(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 210nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116426(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 260nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116423(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ben...)
Affinity DataIC50: 370nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116432(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-f...)
Affinity DataIC50: 410nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116433(4-[1-(Adamantane-1-carbonyl)-piperidin-4-yloxy]-be...)
Affinity DataIC50: 430nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116423(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ben...)
Affinity DataIC50: 530nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116417(4-(1-Diphenylcarbamoyl-piperidin-4-ylidenemethyl)-...)
Affinity DataIC50: 540nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116417(4-(1-Diphenylcarbamoyl-piperidin-4-ylidenemethyl)-...)
Affinity DataIC50: 690nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116420(3-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type 2 of human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116417(4-(1-Diphenylcarbamoyl-piperidin-4-ylidenemethyl)-...)
Affinity DataIC50: 830nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116422(4-[1-(3,3-Diphenyl-propionyl)-piperidin-4-ylidenem...)
Affinity DataIC50: 880nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116428(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-m...)
Affinity DataIC50: 940nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116422(4-[1-(3,3-Diphenyl-propionyl)-piperidin-4-ylidenem...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116432(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-f...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116432(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-f...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116430(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116425(4-(1-Diphenylacetyl-piperidin-4-yloxy)-benzoic aci...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type 2 of human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116422(4-[1-(3,3-Diphenyl-propionyl)-piperidin-4-ylidenem...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116419(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibitory activity against Steroid 5-alpha-reductase type I of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116428(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-m...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116426(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116416(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116419(4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-ylidene...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116424({4-[1-(2,2-Dicyclohexyl-acetyl)-piperidin-4-yliden...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116423(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ben...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Human)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116428(4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-3-m...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 from human benign prostatic hyperplasia (BPH) tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116416(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type 2 of rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116418([4-(1-Diphenylacetyl-piperidin-4-ylidenemethyl)-ph...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Rat)
Saarland University

Curated by ChEMBL
LigandPNGBDBM50116426(4-[1-(Adamantane-1-carbonyl)-piperidin-4-ylideneme...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of Steroid 5-alpha-reductase type I from rat ventral prostate (RVP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed