Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50037187 Sort by
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131992(5-Bromo-3-[2-(4-fluoro-phenyl)-2-oxo-ethylidene]-1...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131998(5-Bromo-3-(2-oxo-2-p-tolyl-ethylidene)-1,3-dihydro...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50154618(cid_5477132 | 5-bromo-3-(2-oxo-2-phenylethylidene)...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50409725(CHEMBL1213804)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131991(CHEMBL126602 | cid_682361 | 3-(2-Oxo-2-phenyl-ethy...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132002(3-(4-Trifluoromethyl-benzylidene)-1,3-dihydro-indo...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM4291(CHEMBL293798 | (2-Oxo-3-indolinidene)malononitrile...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50409725(CHEMBL1213804)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human Cyclin-dependent kinase 1 cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM7266(cid_3820 | NSC 664704 | 9-bromopaullone | 14-bromo...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50131991(CHEMBL126602 | cid_682361 | 3-(2-Oxo-2-phenyl-ethy...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human Cyclin-dependent kinase 1 cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132004(3-(2,6-Dichloro-benzylidene)-1,3-dihydro-indol-2-o...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132005(CHEMBL362785 | 5-methoxy-3-(4-oxo-2-thioxothiazoli...)
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132010(5-Fluoro-3-(4-oxo-2-thioxo-thiazolidin-5-ylidene)-...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132007(3-(piperidin-2-ylmethylene)indolin-2-one | 3-Piper...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131997(2-Cyano-2-(2-oxo-1,2-dihydro-indol-3-ylidene)-acet...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50131992(5-Bromo-3-[2-(4-fluoro-phenyl)-2-oxo-ethylidene]-1...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human Cyclin-dependent kinase 1 cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50131998(5-Bromo-3-(2-oxo-2-p-tolyl-ethylidene)-1,3-dihydro...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human Cyclin-dependent kinase 1 cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50154618(cid_5477132 | 5-bromo-3-(2-oxo-2-phenylethylidene)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Cyclin-dependent kinase 1 cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132003((Z)-1H,1''H-[2,3'']Biindolylidene-3,2''-dione 3-ox...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132009(cid_725903 | CHEMBL127205 | 3-(2-Oxo-propylidene)-...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132006(3-(4-chlorobenzylidene)indolin-2-one | 3-(4-Chloro...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132001(Cyano-(2-oxo-1,2-dihydro-indol-3-ylidene)-acetic a...)
Affinity DataIC50: 4.17E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131995((E)-3-(4-hydroxybenzylidene)indolin-2-one | 3-(4-H...)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50132008(3-(3,3-Dimethyl-2-oxo-butylidene)-1,3-dihydro-indo...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131996(3-Methylaminomethylene-1,3-dihydro-indol-2-one | C...)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50326169((S)-methyl 4-hydroxy-2-(4-hydroxy-3-(3-methylbut-2...)
Affinity DataIC50: 9.40E+4nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50154618(cid_5477132 | 5-bromo-3-(2-oxo-2-phenylethylidene)...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of Plasmodium falciparum cyclin dependent protein kinase, PfPK5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131998(5-Bromo-3-(2-oxo-2-p-tolyl-ethylidene)-1,3-dihydro...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of Plasmodium falciparum cyclin dependent protein kinase, PfPK5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50409725(CHEMBL1213804)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of Plasmodium falciparum cyclin dependent protein kinase, PfPK5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131991(CHEMBL126602 | cid_682361 | 3-(2-Oxo-2-phenyl-ethy...)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of Plasmodium falciparum cyclin dependent protein kinase, PfPK5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM4622(CHEMBL127907 | 3-[(6,7-dimethoxyquinazolin-4-yl)am...)
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50131992(5-Bromo-3-[2-(4-fluoro-phenyl)-2-oxo-ethylidene]-1...)
Affinity DataIC50: 1.90E+5nMAssay Description:Inhibition of Plasmodium falciparum cyclin dependent protein kinase, PfPK5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM5718(2,6,9-Trisubstituted purine deriv. 26 | 2-{[6-(ben...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMO15-related protein kinase Pfmrk(malaria parasite P. falciparum)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against Plasmodium falciparum cyclin dependent protein kinase, PfmrkMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed