Compile Data Set for Download or QSAR
maximum 50k data
Found 64 Enz. Inhib. hit(s) with all data for entry = 50000141
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001778((Lu 23-086)1-(2-{4-[1-(4-Fluoro-phenyl)-1H-indol-3...)
Affinity DataIC50:  0.0820nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001991(1-(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  0.240nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002008(1-(2-{4-[1-(4-Fluoro-phenyl)-5-methyl-1H-indol-3-y...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001990(5-Chloro-1-(4-fluoro-phenyl)-3-(4-methyl-piperazin...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002001(1-(2-{4-[5-Fluoro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002015(5-Chloro-1-(4-fluoro-phenyl)-3-(1-methyl-1,2,3,6-t...)
Affinity DataIC50:  0.530nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001996(5-Fluoro-1-(4-fluoro-phenyl)-3-(1-methyl-1,2,3,6-t...)
Affinity DataIC50:  0.740nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002011(1-(4-Fluoro-phenyl)-3-(1-methyl-1,2,3,6-tetrahydro...)
Affinity DataIC50:  0.760nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002014(1-(2-{4-[1-(4-Fluoro-phenyl)-5-methoxy-1H-indol-3-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002004(1-(3-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001990(5-Chloro-1-(4-fluoro-phenyl)-3-(4-methyl-piperazin...)
Affinity DataIC50:  1nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001997(1-(2-{4-[1-(4-Fluoro-phenyl)-5-trifluoromethyl-1H-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002015(5-Chloro-1-(4-fluoro-phenyl)-3-(1-methyl-1,2,3,6-t...)
Affinity DataIC50:  1.10nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002000(1-(4-Fluoro-phenyl)-3-{1-[2-(2-oxo-imidazolidin-1-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002013(1-(2-{4-[5-Bromo-1-(4-fluoro-phenyl)-1H-indol-3-yl...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001994(2-{4-[1-(4-Fluoro-phenyl)-5-trifluoromethyl-1H-ind...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002010(1-(5-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001989(1-(4-Fluoro-phenyl)-3-(1-methyl-1,2,3,6-tetrahydro...)
Affinity DataIC50:  1.60nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002011(1-(4-Fluoro-phenyl)-3-(1-methyl-1,2,3,6-tetrahydro...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001997(1-(2-{4-[1-(4-Fluoro-phenyl)-5-trifluoromethyl-1H-...)
Affinity DataIC50:  1.90nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001993(1-(4-Fluoro-phenyl)-3-{1-[2-(2-oxo-imidazolidin-1-...)
Affinity DataIC50:  2.10nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002007(1-(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002005(1-(6-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  2.20nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002000(1-(4-Fluoro-phenyl)-3-{1-[2-(2-oxo-imidazolidin-1-...)
Affinity DataIC50:  2.20nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002002(1-(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  2.30nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002005(1-(6-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001994(2-{4-[1-(4-Fluoro-phenyl)-5-trifluoromethyl-1H-ind...)
Affinity DataIC50:  2.60nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001995(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-yl]-...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50019966(2-{4-[(1R,3S)-3-(4-Fluoro-phenyl)-6-trifluoromethy...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001996(5-Fluoro-1-(4-fluoro-phenyl)-3-(1-methyl-1,2,3,6-t...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001993(1-(4-Fluoro-phenyl)-3-{1-[2-(2-oxo-imidazolidin-1-...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002004(1-(3-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  3.40nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002008(1-(2-{4-[1-(4-Fluoro-phenyl)-5-methyl-1H-indol-3-y...)
Affinity DataIC50:  3.70nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002013(1-(2-{4-[5-Bromo-1-(4-fluoro-phenyl)-1H-indol-3-yl...)
Affinity DataIC50:  3.80nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002009(5-Chloro-1-(4-fluoro-phenyl)-3-piperidin-4-yl-1H-i...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)
Affinity DataIC50:  4nMAssay Description:Compound was tested for the inhibition of [3H]-spiperone binding to dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataIC50:  4.10nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002010(1-(5-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  4.20nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002006(1-(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001998(1-(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001995(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-yl]-...)
Affinity DataIC50:  4.5nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002001(1-(2-{4-[5-Fluoro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  4.70nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002003(1-(2-{4-[1-(4-Fluoro-phenyl)-5-methanesulfonyl-1H-...)
Affinity DataIC50:  5.80nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001991(1-(2-{4-[5-Chloro-1-(4-fluoro-phenyl)-1H-indol-3-y...)
Affinity DataIC50:  6.5nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  7.5nMAssay Description:Compound was tested for the inhibition of [3H]-spiperone binding to dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50002003(1-(2-{4-[1-(4-Fluoro-phenyl)-5-methanesulfonyl-1H-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50019966(2-{4-[(1R,3S)-3-(4-Fluoro-phenyl)-6-trifluoromethy...)
Affinity DataIC50:  10nMAssay Description:Tested for the inhibition of [3H]-spiperone binding to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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