Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50037218
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12751(CHEMBL152854 | 1-(3-carbamimidoylphenyl)-3-methyl-...)
Affinity DataKi:  0.0130nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  0.150nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  0.300nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135953(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  0.460nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135943(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  0.540nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135960(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  0.880nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135945(1-[2-(aminomethyl)phenyl]-N-(3-fluoro-2'-sulfamoyl...)
Affinity DataKi:  0.910nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135966(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  1nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135961(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  1.70nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135951(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  1.80nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135954(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  2.40nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135966(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  2.60nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18965(CHEMBL134736 | 1-[3-(aminomethyl)phenyl]-3-methyl-...)
Affinity DataKi:  2.70nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135962(2-(4-Methoxy-phenyl)-5-trifluoromethyl-2H-pyrazole...)
Affinity DataKi:  2.80nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135945(1-[2-(aminomethyl)phenyl]-N-(3-fluoro-2'-sulfamoyl...)
Affinity DataKi:  2.90nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135959(2-(4-Methoxy-phenyl)-5-trifluoromethyl-2H-pyrazole...)
Affinity DataKi:  3.5nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12705(N-[2-fluoro-4-(2-methanesulfonylphenyl)phenyl]-1-(...)
Affinity DataKi:  3.60nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135946(2-(2-Aminomethyl-4-methoxy-phenyl)-5-methyl-2H-pyr...)
Affinity DataKi:  3.80nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135955(2-(4-Methoxy-phenyl)-5-trifluoromethyl-2H-pyrazole...)
Affinity DataKi:  4.20nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135953(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  4.30nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135951(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  4.60nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135965(2-(4-Methoxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi:  5.30nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18971(1-(4-methoxyphenyl)-3-methyl-N-[4-(2-sulfamoylphen...)
Affinity DataKi:  11nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135948(2-(4-Methoxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12751(CHEMBL152854 | 1-(3-carbamimidoylphenyl)-3-methyl-...)
Affinity DataKi:  16nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135947(2-(2-Methylaminomethyl-phenyl)-5-trifluoromethyl-2...)
Affinity DataKi:  28nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135949(2-[2-(Isopropylamino-methyl)-phenyl]-5-trifluorome...)
Affinity DataKi:  38nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135945(1-[2-(aminomethyl)phenyl]-N-(3-fluoro-2'-sulfamoyl...)
Affinity DataKi:  58nMAssay Description:Tested in vitro for inhibition of human plasma KallikrieneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  60nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135957(2-[2-(Benzylamino-methyl)-phenyl]-5-trifluoromethy...)
Affinity DataKi:  61nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetPlasma kallikrein(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  61nMAssay Description:Tested in vitro for inhibition of human plasma KallikrieneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135950(2-(3-Methoxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi:  110nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135942(2-[2-(2-Amino-ethyl)-phenyl]-5-trifluoromethyl-2H-...)
Affinity DataKi:  110nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135956(2-(3-Hydroxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi:  164nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18974(CHEMBL139121 | 3-methyl-1-phenyl-N-[4-(2-sulfamoyl...)
Affinity DataKi:  198nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18965(CHEMBL134736 | 1-[3-(aminomethyl)phenyl]-3-methyl-...)
Affinity DataKi:  250nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135941(2-(3-Aminomethyl-4-methoxy-phenyl)-5-methyl-2H-pyr...)
Affinity DataKi:  270nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12751(CHEMBL152854 | 1-(3-carbamimidoylphenyl)-3-methyl-...)
Affinity DataKi:  300nMAssay Description:In vitro for inhibition of human thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135958(2-[2-(3-Amino-propyl)-phenyl]-5-trifluoromethyl-2H...)
Affinity DataKi:  600nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135964(2-(2-Dimethylaminomethyl-phenyl)-5-trifluoromethyl...)
Affinity DataKi:  800nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135944(2-(4-Hydroxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi:  900nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135963(2-(2-Hydroxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi:  1.20E+3nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135966(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro for inhibition of human thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135952(2-(2-Methoxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi: >1.50E+3nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18974(CHEMBL139121 | 3-methyl-1-phenyl-N-[4-(2-sulfamoyl...)
Affinity DataKi: >1.50E+3nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135956(2-(3-Hydroxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi: >1.50E+3nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135953(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  1.50E+3nMAssay Description:In vitro for inhibition of human thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18971(1-(4-methoxyphenyl)-3-methyl-N-[4-(2-sulfamoylphen...)
Affinity DataKi: >1.50E+3nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135965(2-(4-Methoxy-phenyl)-5-methyl-2H-pyrazole-3-carbox...)
Affinity DataKi: >1.50E+3nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135959(2-(4-Methoxy-phenyl)-5-trifluoromethyl-2H-pyrazole...)
Affinity DataKi: >1.50E+3nMAssay Description:Tested in vitro for inhibition of human trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
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