Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50014381
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141817BDBM50141817([1-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-...)
Affinity DataIC50: 23nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141829BDBM50141829((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141822BDBM50141822((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 54nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141819BDBM50141819((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 63nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141812BDBM50141812(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-2-fluoro-phe...)
Affinity DataIC50: 70nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141813BDBM50141813(1-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-meth...)
Affinity DataIC50: 71nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141823BDBM50141823(2-[(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-...)
Affinity DataIC50: 71nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 83nMAssay Description:Inhibition of vascular endothelial growth factor receptor 2 autophosphorylation in intact cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 88nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141810BDBM50141810((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 100nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 100nMAssay Description:Inhibition of c-Kit autophosphorylation in intact cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141832BDBM50141832((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141821BDBM50141821((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 190nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141816BDBM50141816(1-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-meth...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141814BDBM50141814([4-(6,7-Dimethoxy-quinolin-4-yloxy)-phenyl]-(4-iso...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141824BDBM50141824((4-tert-Butyl-phenyl)-{4-[6-methoxy-7-(2-morpholin...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141811BDBM50141811(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-3-fluoro-phe...)
Affinity DataIC50: 260nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141831BDBM50141831((4-tert-Butyl-phenyl)-{4-[6-methoxy-7-(3-piperidin...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141827BDBM50141827(4-[4-(4-tert-Butyl-phenoxy)-phenoxy]-6,7-dimethoxy...)
Affinity DataIC50: 440nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 480nMAssay Description:Inhibition of PDGF-receptor autophosphorylation in intact cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141826BDBM50141826([4-(6,7-Dimethoxy-quinolin-4-yloxy)-phenyl]-(4-met...)
Affinity DataIC50: 780nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141830BDBM50141830(4-[4-(4-tert-Butyl-benzyl)-phenoxy]-6,7-dimethoxy-...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141828BDBM50141828((4-tert-Butyl-cyclohexyl)-[4-(6,7-dimethoxy-quinol...)
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141808BDBM50141808(Biphenyl-4-yl-[4-(6,7-dimethoxy-quinolin-4-yloxy)-...)
Affinity DataIC50: 4.60E+3nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141825BDBM50141825([4-(6,7-Dimethoxy-quinolin-4-yloxy)-phenyl]-phenyl...)
Affinity DataIC50: 8.90E+3nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141815BDBM50141815((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGF-receptor autophosphorylation in intact cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of c-Met autophosphorylation of in intact cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInsulin-like growth factor 1 receptor(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141809BDBM50141809(2-(2-{4-[4-(4-tert-Butyl-phenylamino)-phenoxy]-6-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of IGF-receptor 1 autophosphorylation in intact cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141818BDBM50141818(Biphenyl-3-yl-[4-(6,7-dimethoxy-quinolin-4-yloxy)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Kirin Brewery

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50141820BDBM50141820((4-tert-Butyl-phenyl)-[4-(6,7-dimethoxy-quinolin-4...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition against autophosphorylation of Fibroblast growth factor receptor 2 in the human scirrhous gastric carcinoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed