Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50022505
Affinity DataIC50: 86nMAssay Description:Inhibition of human IGF-IR in mouse NWT-21 cells assessed as inhibition of autophosphorylation of IGF-IR at pH 7.2 incubated for 90 mins followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibition of IGF-IR in human MCF7 cells assessed as inhibition of anchorage-independent growth incubated for 30 mins and measured after 3 weeks by c...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of GST tagged human Ins-R expressed in baculovirus at pH 7.6 measured after 20 mins in presence of gamma-[33P]-ATP by scintillation counte...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of GST tagged human IGF-IR expressed in baculovirus at pH 7.6 measured after 20 mins in presence of gamma-[33P]-ATP by scintillation count...More data for this Ligand-Target Pair
Affinity DataIC50: 162nMAssay Description:Inhibition of IGF-IR in human MCF7 cells expressing IGF-I assessed as cell survival in the absence of serum incubated for 72 hrs by MTS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of GST tagged human Flt-3 expressed in baculovirus at pH 7.6 measured after 15 mins in presence of gamma-[33P]-ATP by scintillation counte...More data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibition of GST tagged Tek (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP by scint...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of GST tagged Flt-1 (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP by sci...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of GST tagged human HER-4 expressed in baculovirus at pH 7.5 measured after 15 mins in presence of gamma-[33P]-ATP by scintillation counte...More data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of human IGF-IR expressed in mouse NWT-21 cells assessed as inhibition of proliferative capacity incubated for 72 hrs in presence of serum...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST tagged PDGFR-beta (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP b...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of GST tagged KDR (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP by scint...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Ins-R in A14 [Human melanoma] cells assessed as inhibition of autophosphorylation of Ins-R incubated for 90 mins followed by insulin st...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of GST tagged chicken c-Src expressed in baculovirus at pH 7.5 measured after 10 mins in presence of gamma-[33P]-ATP by scintillation coun...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of GST tagged human Flt-4 expressed in baculovirus at pH 7.6 measured after 15 mins in presence of gamma-[33P]-ATP by scintillation counte...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of GST tagged c-Kit (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP by sci...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of GST tagged c-Met (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP by sci...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of GST tagged FGFR-1 (unknown origin) expressed in baculovirus at pH 7.6 measured after 10 to 30 mins in presence of gamma-[33P]-ATP by sc...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of GST tagged human HER-2 expressed in baculovirus at pH 7.5 measured after 15 mins in presence of gamma-[33P]-ATP by scintillation counte...More data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PDK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of c-Kit (unknown origin) in human GIST882 cells assessed as inhibition of autophosphorylation of c-Kit incubated for 90 mins in presence ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of GST tagged human HER-1 expressed in baculovirus at pH 7.5 measured after 15 mins in presence of gamma-[33P]-ATP by scintillation counte...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST tagged c-Abl (unknown origin) expressed in baculovirus infected Sf9 cells at pH 7.5 measured after 10 mins in presence of gamma-[33...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged c-Raf-1 (unknown origin) expressed in baculovirus infected in Sf21 cells at pH 7.5 measured after 30 mins in presence of gam...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PKB expressed in baculovirus at pH 7.2 measured after 30 mins in presence of gamma-[33P]-ATP by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Bcr-Abl (unknown origin) in mouse 32D cells assessed as inhibition of autophosphorylation of Bcr-Abl incubated for 90 mins in presence ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HER-1 in human A-431 cells assessed as inhibition of autophosphorylation of HER-1 incubated for 90 mins followed by EGF stimulation mea...More data for this Ligand-Target Pair
