Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50014795
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147513BDBM50147513(2-[3-[5-(4-Chloro-phenyl)-benzooxazol-2-yl]-4-(2-m...)
Affinity DataIC50: 200nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147546BDBM50147546(2-[3-(5-Benzo[1,3]dioxol-5-yl-benzooxazol-2-yl)-4-...)
Affinity DataIC50: 200nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147534BDBM50147534(1,3-dioxo-2-(3-(5-phenylbenzo[d]oxazol-2-yl)-4-(pr...)
Affinity DataIC50: 250nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147544BDBM50147544(2-(2-methoxy-5-(5-(4-(trifluoromethoxy)phenyl)benz...)
Affinity DataIC50: 400nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147533BDBM50147533(2-(5-(5-(3,5-difluorophenyl)benzo[d]oxazol-2-yl)-2...)
Affinity DataIC50: 400nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147537BDBM50147537(2-{5-[5-(4-Fluoro-phenyl)-benzooxazol-2-yl]-2-meth...)
Affinity DataIC50: 400nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147522BDBM50147522(2-[4-Butylamino-3-(5-phenyl-benzooxazol-2-yl)-phen...)
Affinity DataIC50: 400nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147539BDBM50147539(2-(2-methoxy-5-(5-(4-methoxyphenyl)benzo[d]oxazol-...)
Affinity DataIC50: 450nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147517BDBM50147517(2-[3-[5-(4-Fluoro-phenyl)-benzooxazol-2-yl]-4-(2-m...)
Affinity DataIC50: 500nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147528BDBM50147528(2-(5-(5-(3,4-difluorophenyl)benzo[d]oxazol-2-yl)-2...)
Affinity DataIC50: 600nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147536BDBM50147536(2-(5-(5-(3-chlorophenyl)benzo[d]oxazol-2-yl)-2-met...)
Affinity DataIC50: 600nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147535BDBM50147535(2-(5-(5-(benzo[d][1,3]dioxol-5-yl)benzo[d]oxazol-2...)
Affinity DataIC50: 750nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147519BDBM50147519(2-{5-[5-(2,4-Difluoro-phenyl)-benzooxazol-2-yl]-2-...)
Affinity DataIC50: 800nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147518BDBM50147518(2-{4-(2-Methoxy-ethylamino)-3-[5-(4-trifluorometho...)
Affinity DataIC50: 800nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147530BDBM50147530(2-(3-(5-(3,5-difluorophenyl)benzo[d]oxazol-2-yl)-4...)
Affinity DataIC50: 900nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147510BDBM50147510(2-[4-Ethylamino-3-(5-phenyl-benzooxazol-2-yl)-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147531BDBM50147531(2-(5-(5-(3-fluorophenyl)benzo[d]oxazol-2-yl)-2-met...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147538BDBM50147538(2-[4-Ethoxy-3-(5-phenyl-benzooxazol-2-yl)-phenyl]-...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147515BDBM50147515(2-[3-(5-Chloro-benzooxazol-2-yl)-phenyl]-1,3-dioxo...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147509BDBM50147509(2-{4-(2-Methoxy-ethylamino)-3-[5-(4-trifluoromethy...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147511BDBM50147511(2-[3-[5-(3-Chloro-4-fluoro-phenyl)-benzooxazol-2-y...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147524BDBM50147524(2-(4-(2-methoxyethylamino)-3-(5-phenylbenzo[d]oxaz...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147527BDBM50147527(2-[3-(5-Methyl-benzooxazol-2-yl)-phenyl]-1,3-dioxo...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147506BDBM50147506(2-(3-(5-(4-chlorophenyl)benzo[d]oxazol-2-yl)-4-met...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147548BDBM50147548(2-[3-[5-(3-Chloro-phenyl)-benzooxazol-2-yl]-4-(2-m...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147516BDBM50147516(2-[2-Ethoxy-5-(5-phenyl-benzooxazol-2-yl)-phenyl]-...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147521BDBM50147521(1,3-Dioxo-2-[3-(5-phenyl-benzooxazol-2-yl)-phenyl]...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147551BDBM50147551(2-{5-[5-(3-Cyano-phenyl)-benzooxazol-2-yl]-2-metho...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147523BDBM50147523(2-{2-Methoxy-5-[5-(3-methoxy-phenyl)-benzooxazol-2...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147529BDBM50147529(2-[3-[5-(3,5-Difluoro-phenyl)-benzooxazol-2-yl]-4-...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147525BDBM50147525(2-(5-(5-chlorobenzo[d]oxazol-2-yl)-2-methoxyphenyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147549BDBM50147549(2-[2-Methoxy-5-(5-phenyl-benzooxazol-2-yl)-phenyl]...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147514BDBM50147514(2-(4-isopropoxy-3-(5-phenylbenzo[d]oxazol-2-yl)phe...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147545BDBM50147545(2-[2-(2-Methoxy-ethoxy)-5-(5-phenyl-benzooxazol-2-...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147540BDBM50147540(2-{5-[5-(4-Chloro-phenyl)-benzooxazol-2-yl]-2-meth...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147520BDBM50147520(2-[4-(2-Methoxy-ethoxy)-3-(5-phenyl-benzooxazol-2-...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147512BDBM50147512(2-(4-(methyl(propyl)amino)-3-(5-phenylbenzo[d]oxaz...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147526BDBM50147526(2-(3-Benzooxazol-2-yl-phenyl)-1,3-dioxo-indan-5-ca...)
Affinity DataIC50: 8.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147508BDBM50147508(2-(2-methoxy-5-(5-(2-methoxyphenyl)benzo[d]oxazol-...)
Affinity DataIC50: 9.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147547BDBM50147547(2-(5-(5-(3-acetamidophenyl)benzo[d]oxazol-2-yl)-2-...)
Affinity DataIC50: 9.00E+3nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147532BDBM50147532(2-[4-Methylamino-3-(5-phenyl-benzooxazol-2-yl)-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147541BDBM50147541(2-{4-Methoxy-3-[5-(4-trifluoromethoxy-phenyl)-benz...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147543BDBM50147543(2-(5-Benzooxazol-2-yl-2-methoxy-phenyl)-1,3-dioxo-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147550BDBM50147550(2-[4-tert-Butoxy-3-(5-phenyl-benzooxazol-2-yl)-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147542BDBM50147542(2-[4-(2-Dimethylamino-ethoxy)-3-(5-phenyl-benzooxa...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50147507BDBM50147507(2-[2-Methoxy-5-(5-methyl-benzooxazol-2-yl)-phenyl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vivo inhibitory activity against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed