Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50016462
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169361BDBM50169361(3-(3-Cyclobutyl-2-oxo-2,3-dihydro-1H-benzoimidazol...)
Affinity DataIC50: 3.30nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169346BDBM50169346(5-(3-Isopropyl-2-oxo-2,3-dihydro-1H-benzoimidazol-...)
Affinity DataIC50: 4.70nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169354BDBM50169354(5-(3-cyclopentyl-2-oxo-2,3-dihydro-1H-benzimidazol...)
Affinity DataIC50: 5.60nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169352BDBM50169352(3-(3-Cyclopentyl-2-oxo-2,3-dihydro-1H-benzoimidazo...)
Affinity DataIC50: 5.70nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219259BDBM50219259(5-(3-cyclobutyl-2-oxo-2,3-dihydro-1H-benzimidazol-...)
Affinity DataIC50: 10.9nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169355BDBM50169355(1-Methyl-5-(2-oxo-3-pentyl-2,3-dihydro-1H-benzoimi...)
Affinity DataIC50: 11.7nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169359BDBM50169359(5-(3-Isopropyl-2-oxo-2,3-dihydro-1H-benzoimidazol-...)
Affinity DataIC50: 24.8nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169345BDBM50169345(3-Fluoro-5-(2-oxo-3-pentyl-2,3-dihydro-1H-benzoimi...)
Affinity DataIC50: 29nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169340BDBM50169340(3-Fluoro-5-(3-isopropyl-2-oxo-2,3-dihydro-1H-benzo...)
Affinity DataIC50: 29.6nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169358BDBM50169358(2-Fluoro-5-(3-isopropyl-2-oxo-2,3-dihydro-1H-benzo...)
Affinity DataIC50: 60.3nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169350BDBM50169350(6-(3-Fluoro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...)
Affinity DataIC50: 77.9nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169341BDBM50169341(3-(3-Cyclohexyl-2-oxo-2,3-dihydro-1H-benzoimidazol...)
Affinity DataIC50: 83.6nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169357BDBM50169357(1-Cyclopentyl-6-(3,4-difluoro-phenyl)-1,3-dihydro-...)
Affinity DataIC50: 96.8nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169344BDBM50169344(6-(3,5-Dichloro-phenyl)-1-isopropyl-1,3-dihydro-be...)
Affinity DataIC50: 100nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169343BDBM50169343(6-(3-Chloro-4-fluoro-phenyl)-1-isopropyl-1,3-dihyd...)
Affinity DataIC50: 106nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169348BDBM50169348(6-(3-Chloro-4-fluoro-phenyl)-1-cyclobutyl-1,3-dihy...)
Affinity DataIC50: 106nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169342BDBM50169342(6-(3-Chloro-4-fluoro-phenyl)-1-cyclopentyl-1,3-dih...)
Affinity DataIC50: 135nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169363BDBM50169363(3-Fluoro-5-(2-oxo-3-phenyl-2,3-dihydro-1H-benzoimi...)
Affinity DataIC50: 137nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169349BDBM50169349(1-Cyclobutyl-6-(3,4-difluoro-phenyl)-1,3-dihydro-b...)
Affinity DataIC50: 175nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169356BDBM50169356(6-(3,4-Difluoro-phenyl)-1-isopropyl-1,3-dihydro-be...)
Affinity DataIC50: 207nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169347BDBM50169347(6-(4-Fluoro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...)
Affinity DataIC50: 295nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169362BDBM50169362(6-(2-Fluoro-phenyl)-1-isopropyl-1,3-dihydro-benzoi...)
Affinity DataIC50: 412nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169360BDBM50169360(6-(3-Chloro-4-fluoro-phenyl)-1-pentyl-1,3-dihydro-...)
Affinity DataIC50: 426nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50169353BDBM50169353(3-[3-(3-Chloro-phenyl)-2-oxo-2,3-dihydro-1H-benzoi...)
Affinity DataIC50: 3.00E+3nMAssay Description:Progesterone receptor agonist activity in human T47D breast carcinoma cell alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed