Compile Data Set for Download or QSAR
Report error Found 95 Enz. Inhib. hit(s) with all data for entry = 50003763
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475680BDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  87nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475680BDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  851nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475680BDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  933nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475680BDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  977nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004656BDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  1.23E+3nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475680BDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  1.23E+3nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475675BDBM50475675(CHEMBL380759)
Affinity DataKi:  1.95E+3nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475675BDBM50475675(CHEMBL380759)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475675BDBM50475675(CHEMBL380759)
Affinity DataKi:  3.24E+3nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475675BDBM50475675(CHEMBL380759)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004656BDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  6.31E+3nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475675BDBM50475675(CHEMBL380759)
Affinity DataKi:  9.12E+3nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475683BDBM50475683(CHEMBL2092820)
Affinity DataKi:  9.33E+3nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475678BDBM50475678(CHEMBL2093084)
Affinity DataKi:  1.55E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475679BDBM50475679(CHEMBL2093082)
Affinity DataKi:  2.88E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475679BDBM50475679(CHEMBL2093082)
Affinity DataKi:  2.88E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475678BDBM50475678(CHEMBL2093084)
Affinity DataKi:  3.39E+4nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475678BDBM50475678(CHEMBL2093084)
Affinity DataKi:  3.39E+4nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004656BDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  3.80E+4nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004656BDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  4.37E+4nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475678BDBM50475678(CHEMBL2093084)
Affinity DataKi:  4.68E+4nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475676BDBM50475676(CHEMBL2092736)
Affinity DataKi:  5.13E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475679BDBM50475679(CHEMBL2093082)
Affinity DataKi:  5.75E+4nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004656BDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  6.92E+4nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475687BDBM50475687(CHEMBL2092735)
Affinity DataKi:  7.76E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475688BDBM50475688(CHEMBL2092737)
Affinity DataKi:  8.71E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475677BDBM50475677(CHEMBL3351105)
Affinity DataKi:  8.91E+4nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475678BDBM50475678(CHEMBL2093084)
Affinity DataKi:  9.33E+4nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475681BDBM50475681(CHEMBL3351103)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475684BDBM50475684(CHEMBL3350064)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475685BDBM50475685(CHEMBL2093083)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475681BDBM50475681(CHEMBL3351103)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475682BDBM50475682(CHEMBL3350063)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475683BDBM50475683(CHEMBL2092820)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475679BDBM50475679(CHEMBL2093082)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475674BDBM50475674(CHEMBL3350062)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475676BDBM50475676(CHEMBL2092736)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475677BDBM50475677(CHEMBL3351105)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475683BDBM50475683(CHEMBL2092820)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475684BDBM50475684(CHEMBL3350064)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475684BDBM50475684(CHEMBL3350064)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475681BDBM50475681(CHEMBL3351103)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475682BDBM50475682(CHEMBL3350063)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475676BDBM50475676(CHEMBL2092736)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475674BDBM50475674(CHEMBL3350062)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475686BDBM50475686(CHEMBL3351104)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475679BDBM50475679(CHEMBL2093082)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475686BDBM50475686(CHEMBL3351104)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475683BDBM50475683(CHEMBL2092820)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Florence

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50475676BDBM50475676(CHEMBL2092736)
Affinity DataKi: <1.00E+5nMAssay Description:Binding affinity to cloned human muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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