Compile Data Set for Download or QSAR
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Found 20 Enz. Inhib. hit(s) with all data for entry = 50017592
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  12nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  16nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  17nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  200nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  250nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  290nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  380nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  430nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  440nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: >4.10E+3nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184346((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184348((Z)-4-[6-((Z)-3-ethoxycarbonyl-3-hydroxy-acryloyl)...)
Affinity DataIC50: >3.33E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed