TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against MDR human HL60R cell lineMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antiproliferative activity against human K562 cell line expressing Bcr-AblMore data for this Ligand-Target Pair