Compile Data Set for Download or QSAR
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Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50037718
LigandPNGBDBM50191431(5-bromoindirubin-3'-oxime | CHEMBL379494)
Affinity DataIC50:  28nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  83nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50132003((Z)-1H,1''H-[2,3'']Biindolylidene-3,2''-dione 3-ox...)
Affinity DataIC50:  100nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191421(3-(3-(methoxyimino)indolin-2-ylidene)indolin-2-one...)
Affinity DataIC50:  400nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191448((2'Z,3'E)-7-fluoroindirubin-3'-oxime | CHEMBL21217...)
Affinity DataIC50:  510nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191394(2,3'-biindole-2',3(1H,1'H)-dione 3-(O-acetyloxime)...)
Affinity DataIC50:  700nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191420((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-piperazin-1-yl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191436((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-piperazin-1-yl...)
Affinity DataIC50:  5.40E+3nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191418((2'Z,3'E)-7-chloroindirubin-3'-oxime | CHEMBL21365...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191430((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-morph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191435((2'Z,3'E)-1-Methyl-7-bromoindirubin-3'-[O-(2-imida...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191401((2'Z,3' E)-1-methyl-7-bromoindirubin-3'-[O-(2-pyrr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191447((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-diethylaminoet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191415((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-pyrrolidin-1-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191429((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-diethylaminoet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191444((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(N,Ndiet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191426((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-imidazol-1-yle...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191446((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-morpholin-1-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191411((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-dimethylaminoe...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191404((2'Z, 3'E)-7-bromoindirubin-3'-[O-(2-pyrrolidin-1-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191426((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-imidazol-1-yle...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191420((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-piperazin-1-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191436((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-piperazin-1-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191403((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-dieth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191437((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-morpholin-1-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191429((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-diethylaminoet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191400((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-bromo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191395((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-pyrro...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191428((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-morph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191399((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-dieth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191422((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-dimet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50349806(INDIRUBIN)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191396((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-dimethylaminoe...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191402((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-dimet...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191401((2'Z,3' E)-1-methyl-7-bromoindirubin-3'-[O-(2-pyrr...)
Affinity DataIC50:  1.30E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191395((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-pyrro...)
Affinity DataIC50:  1.88E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191405((2'Z,3'E)-7-bromoindirubin-3'-oxime | CHEMBL373834)
Affinity DataIC50:  2.00E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191422((2'Z,3'E)-1-methyl-7-bromoindirubin-3'-[O-(2-dimet...)
Affinity DataIC50:  2.40E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191438((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-bromoethyl)oxi...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191396((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-dimethylaminoe...)
Affinity DataIC50:  2.50E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191415((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-pyrrolidin-1-y...)
Affinity DataIC50: >3.00E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAryl hydrocarbon receptor(Human)
Cnrs

Curated by ChEMBL
LigandPNGBDBM50191411((2'Z,3'E)-7-bromoindirubin-3'-[O-(2-dimethylaminoe...)
Affinity DataIC50: >3.00E+4nMAssay Description:Survival of mouse AhR +/+ 5L cells after 48 hrs by MTS reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191405((2'Z,3'E)-7-bromoindirubin-3'-oxime | CHEMBL373834)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191398((2'Z,3'E)-7-iodoindirubin-3'-oxime | CHEMBL209648)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191412((2'Z,3'E)-7-iodo-1-methylindirubin-3'-oxime | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191409((2'Z,3'E)-7-chloro-1-methylindirubin-3'-acetoxime ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191410((Z)-1'-Methyl-1H,1'H-[2,3']biindolylidene-3,2'-dio...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191417((2'Z,3'E)-7-iodoindirubin-3'-methoxime | CHEMBL213...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191423((2'Z,3'E)-7-bromoindirubin-3'-[O-(N,N-diethylcarba...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50191392((2'Z,3'E)-7-bromo-1-methylindirubin-3'-acetoxime |...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mammalian CDK5/p25More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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