Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50037891
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212652(CHEMBL375468 | N-methyl-3-[(4-phenoxyphenyl)oxy]pr...)
Affinity DataEC50:  370nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212678(CHEMBL229075 | N,N-dimethyl-3-[(4-phenoxyphenyl)ox...)
Affinity DataEC50:  464nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212654(5-(4-phenoxybenzamido)pentylamine hydrochloride | ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212656(3-[(4-phenoxyphenyl)oxy]propylamine hydrochloride ...)
Affinity DataEC50:  433nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212657(7-phenoxy-1-phenyl-2,3,4,5-tetrahydro-3-benzazepin...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212655(CHEMBL375470 | N,N-dimethyl-5-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212658(2-(1-phenoxynaphthalen-4-yl)-2-phenylethylamine hy...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212659(2-(1-hydroxynaphthalen-4-yl)-2-phenylethylamine hy...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212653(2-(4-phenoxyphenyl)but-3-yn-1-amine hydrochloride ...)
Affinity DataEC50:  929nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212660(8-phenoxy-1-phenyl-2,3,4,5-tetrahydro-3-benzazepin...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212661(2-(1-phenoxynaphthalen-4-yl)ethylamine | CHEMBL229...)
Affinity DataEC50:  26nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212662(2-(4-phenoxyphenyl)-4-phenylbut-3-yn-1-amine hydro...)
Affinity DataEC50:  41nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212663(3-(4-phenoxybenzamido)propylamine hydrochloride | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212662(2-(4-phenoxyphenyl)-4-phenylbut-3-yn-1-amine hydro...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212657(7-phenoxy-1-phenyl-2,3,4,5-tetrahydro-3-benzazepin...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212660(8-phenoxy-1-phenyl-2,3,4,5-tetrahydro-3-benzazepin...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212664(CHEMBL229185 | N,N-dimethyl-3-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212652(CHEMBL375468 | N-methyl-3-[(4-phenoxyphenyl)oxy]pr...)
Affinity DataEC50:  66nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212665(2-(4-phenoxyphenyl)ethanaminium chloride | CHEMBL2...)
Affinity DataEC50:  420nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212666(CHEMBL375469 | N,N-dimethyl-2-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212669(2-(4-(4-hydroxyphenoxy)-3-iodophenyl)ethanaminium ...)
Affinity DataEC50:  33nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212667(2-(4-phenoxybenzamido)ethylamine hydrochloride | C...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212668(3-[(3-phenoxyphenyl)oxy]propylamine hydrochloride ...)
Affinity DataEC50:  373nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212670(4-(4-phenoxybenzamido)butylamine hydrochloride | C...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212673(2-(1-methoxynaphthalen-4-yl)-2-phenylethylamine hy...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212671(2-(3-phenoxyphenyl)-2-phenylethylamine hydrochlori...)
Affinity DataEC50:  19nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212672(CHEMBL229234 | N,N-dimethyl-4-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212656(3-[(4-phenoxyphenyl)oxy]propylamine hydrochloride ...)
Affinity DataEC50:  758nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212674(2-(4-phenoxyphenyl)-2-phenylethylamine hydrochlori...)
Affinity DataEC50:  28nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212659(2-(1-hydroxynaphthalen-4-yl)-2-phenylethylamine hy...)
Affinity DataEC50:  716nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212675(2-methyl-2-(4-phenoxyphenyl)propan-1-amine hydroch...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212672(CHEMBL229234 | N,N-dimethyl-4-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212661(2-(1-phenoxynaphthalen-4-yl)ethylamine | CHEMBL229...)
Affinity DataEC50:  101nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212676(2-(4-phenoxyphenyl)-3-phenylpropan-1-amine hydroch...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212671(2-(3-phenoxyphenyl)-2-phenylethylamine hydrochlori...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212677(2-(4-phenoxyphenyl)propan-1-amine hydrochloride | ...)
Affinity DataEC50:  250nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212668(3-[(3-phenoxyphenyl)oxy]propylamine hydrochloride ...)
Affinity DataEC50:  885nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212665(2-(4-phenoxyphenyl)ethanaminium chloride | CHEMBL2...)
Affinity DataEC50:  63nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212667(2-(4-phenoxybenzamido)ethylamine hydrochloride | C...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212664(CHEMBL229185 | N,N-dimethyl-3-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212676(2-(4-phenoxyphenyl)-3-phenylpropan-1-amine hydroch...)
Affinity DataEC50:  140nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212670(4-(4-phenoxybenzamido)butylamine hydrochloride | C...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212674(2-(4-phenoxyphenyl)-2-phenylethylamine hydrochlori...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212654(5-(4-phenoxybenzamido)pentylamine hydrochloride | ...)
Affinity DataEC50:  905nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212658(2-(1-phenoxynaphthalen-4-yl)-2-phenylethylamine hy...)
Affinity DataEC50:  52nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212655(CHEMBL375470 | N,N-dimethyl-5-(4-phenoxybenzamido)...)
Affinity DataEC50:  109nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212663(3-(4-phenoxybenzamido)propylamine hydrochloride | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Mus musculus (Mouse))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212666(CHEMBL375469 | N,N-dimethyl-2-(4-phenoxybenzamido)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at mouse TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212673(2-(1-methoxynaphthalen-4-yl)-2-phenylethylamine hy...)
Affinity DataEC50:  270nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrace amine-associated receptor 1(Rattus norvegicus (Rat))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50212678(CHEMBL229075 | N,N-dimethyl-3-[(4-phenoxyphenyl)ox...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at rat TAAR1 expressed in HEK293 cells assessed as cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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