Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50004000
TargetSodium-dependent dopamine transporter(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478609(Hydroperoxycadiforin)
Affinity DataIC50: 64.7nMAssay Description:Inhibition of dopamine uptake at DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478609(Hydroperoxycadiforin)
Affinity DataIC50: 64.7nMAssay Description:Inhibition of noradrenaline transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478609(Hydroperoxycadiforin)
Affinity DataIC50: 64.7nMAssay Description:Inhibition of serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478610(CHEMBL479210)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of cyclooxygenase-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50334064((1S,2R,5R,6R,9R,10R,13S,15S)-5-[(2R,3E,5R)-5,6-dim...)
Affinity DataIC50: 3.49E+4nMAssay Description:Inhibition of rat lens aldose reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478610(CHEMBL479210)
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of cyclooxygenase-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 5.57E+4nMAssay Description:Antagonist activity at protein kinase C deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 7.27E+4nMAssay Description:Antagonist activity at protein kinase C epsilonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 8.72E+4nMAssay Description:Antagonist activity at protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 1.04E+5nMAssay Description:Antagonist activity at protein kinase C zetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 1.18E+5nMAssay Description:Antagonist activity at protein kinase C beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 1.18E+5nMAssay Description:Antagonist activity at protein kinase C beta-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Human)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: 3.63E+5nMAssay Description:Antagonist activity at protein kinase C gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed