Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50004000
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478609(Hydroperoxycadiforin)
Affinity DataIC50:  64.7nMAssay Description:Inhibition of dopamine uptake at DATMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478609(Hydroperoxycadiforin)
Affinity DataIC50:  64.7nMAssay Description:Inhibition of noradrenaline transporterMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478609(Hydroperoxycadiforin)
Affinity DataIC50:  64.7nMAssay Description:Inhibition of serotonin transporterMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478610(CHEMBL479210)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of cyclooxygenase-2More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50334064((1S,2R,5R,6R,9R,10R,13S,15S)-5-[(2R,3E,5R)-5,6-dim...)
Affinity DataIC50:  3.49E+4nMAssay Description:Inhibition of rat lens aldose reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478610(CHEMBL479210)
Affinity DataIC50:  4.37E+4nMAssay Description:Inhibition of cyclooxygenase-1More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50:  5.57E+4nMAssay Description:Antagonist activity at protein kinase C deltaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50:  7.27E+4nMAssay Description:Antagonist activity at protein kinase C epsilonMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50:  8.72E+4nMAssay Description:Antagonist activity at protein kinase C alphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50:  1.04E+5nMAssay Description:Antagonist activity at protein kinase C zetaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50:  1.18E+5nMAssay Description:Antagonist activity at protein kinase C beta2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50:  1.18E+5nMAssay Description:Antagonist activity at protein kinase C beta-1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50478505(Chondrillin)
Affinity DataIC50: >3.63E+5nMAssay Description:Antagonist activity at protein kinase C gammaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed