Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50035924
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataKi:  0.450nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50368159(CHEMBL610402 | CHEMBL315056)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50368160(CHEMBL610407)
Affinity DataKi:  7.60nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM42467(N6-PHENYLADENOSINE | cid_101430 | (2R,3R,4S,5R)-2-...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50449718(CHEMBL312917)
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  50nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50009525(2-CI Adenosine | 2-Chloroadenosine | CHEMBL285819 ...)
Affinity DataKi:  76nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50118810(CHEMBL139000 | N6-[(R)-1-Methyl-2-phenylethyl]ado ...)
Affinity DataKi:  220nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50368159(CHEMBL610402 | CHEMBL315056)
Affinity DataKi:  220nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM25400(cid_657378 | CPA | CHEMBL68738 | (2R,3R,4S,5R)-2-[...)
Affinity DataKi:  510nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataKi:  950nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM42467(N6-PHENYLADENOSINE | cid_101430 | (2R,3R,4S,5R)-2-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50368160(CHEMBL610407)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50080398(N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) | CHEMB...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
University of South Florida

Curated by ChEMBL
LigandPNGBDBM50449718(CHEMBL312917)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed